SCHEMBL19260814

SCHEMBL19260814

NC(=O)c1cc(-c2ccccc2F)c(F)cn1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 8/20 0.52
SCN9A Q15858 2/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
HTR5A P47898 1/20 0.43
CDC7 O00311 1/20 0.43
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
PARP1 P09874 2/20 0.42
PDE4B Q07343 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14877992 0.75 BCAT2 (0.53) GRM2NPC1RAB9APARP1
SCHEMBL29777916 0.73 NPC1 (0.46) GRM2NPC1RAB9ACDC7ALOX5AP
SCHEMBL2113823 0.73 NPC1 (0.59) GRM2NPC1RAB9ACDC7ALOX5AP
SCHEMBL19659747 0.72 GRM2 (0.44) GRM2SCN9ANPC1RAB9ACDC7
SCHEMBL18036225 0.72 KDM4E (0.44) GRM2CDC7ALOX5APFEN1
SCHEMBL31341112 0.71 CDC7 (0.45) NPC1RAB9ACDC7PARP1
SCHEMBL30140611 0.71 NPC1 (0.50) GRM2NPC1RAB9A
SCHEMBL6634187 0.70 SIRT6 (0.50) GRM2
SCHEMBL16318634 0.70 KDM4E (0.43) GRM2NPC1RAB9A
SCHEMBL5285579 0.70 MAPT (0.47) GRM2NPC1RAB9ACDC7PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3416648-A1 PROCESSES FOR THE PREPARATION OF A BACE INHIBITOR Merck Sharp & Dohme Corp. (US) 2018-12-26 EP disclosed
WO-2017142804-A1 PROCESSES FOR THE PREPARATION OF A BACE INHIBITOR MERCK SHARP & DOHME CORP. (US) 2017-08-24 WO disclosed