SCHEMBL1929065

SCHEMBL1929065

CCOC(=O)[C@@H]1CCCCN1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.44
SLC6A3 Q01959 3/20 0.44
SLC6A4 P31645 2/20 0.44
ALDH1A1 P00352 2/20 0.41
PRCP P42785 1/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PPM1B O75688 1/20 0.38
PTPN1 P18031 1/20 0.38
PPP1CC P36873 1/20 0.38
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL135813 1.00 SLC6A2 (0.44) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
SCHEMBL3164291 1.00 SLC6A2 (0.44) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
Hydrochloric Acid SCHEMBL6733273 0.98 SLC6A2 (0.46) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
SCHEMBL5429881 0.98 ALDH1A1 (0.44) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
Hydrochloric Acid SCHEMBL6954164 0.98 SLC6A2 (0.46) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
SCHEMBL9438838 0.98 ALDH1A1 (0.44) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
SCHEMBL9438970 0.98 ALDH1A1 (0.44) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
Hydrochloric Acid SCHEMBL1282288 0.98 SLC6A2 (0.46) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
SCHEMBL9439436 0.98 ALDH1A1 (0.44) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP
Oxalic Acid SCHEMBL29060702 0.95 SLC6A2 (0.45) SLC6A2SLC6A3SLC6A4ALDH1A1PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250326732-A1 CHROMEN-2-ONE MODULATORS OF POLRMT PRETZEL THERAPEUTICS, INC. (US) 2025-10-23 US disclosed
WO-2023034346-A1 CHROMEN-2-ONE MODULATORS OF POLRMT PRETZEL THERAPEUTICS, INC. (US) 2023-03-09 WO disclosed
EP-2831069-B1 ISOXAZOLE BETA-LACTAMASE INHIBITORS MERCK SHARP & DOHME (US) 2017-07-12 EP disclosed
US-8436183-B2 Synthetic multimerizing agents ARIAD PHARMACEUTICALS, INC. (US) 2013-05-07 US disclosed
US-8436183-B2 Synthetic multimerizing agents ARIAD PHARMACEUTICALS, INC. (US) 2013-05-07 US disclosed
WO-2013007371-A2 KINETIC RESOLUTION OF CHIRAL AMINES ETH ZURICH (CH) 2013-01-17 WO disclosed
US-20120130076-A1 Synthetic Multimerizing Agents ARIAD PHARMACEUTICALS, INC. (US) 2012-05-24 US disclosed
US-8106191-B2 Compounds based on N- acyl-pipecolyl and N-acyl-prolyl ligand moieties for multimerizing chimeric proteins containing immunophilin-derived domains ARIAD PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed
US-20110152234-A1 Novel Compounds ASTRAZENECA AB (SE) 2011-06-23 US disclosed
US-7956084-B2 Phenyl thiophene carboxamide compounds as inhibitors of the enzyme IKK-2 ASTRAZENECA AB (SE) 2011-06-07 US disclosed
WO-2003010158-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2003-02-06 WO disclosed
EP-0820451-B1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK AS (DK) 2003-01-15 EP disclosed
CN-1315951-A FKBP inhibitors PFIZER LTD (US) 2001-10-03 CN disclosed
US-6239148-B1 TREATMENT OF PAINFUL, HYPERALGESIC AND/OR INFLAMMATORY CONDITIONS IN WHICH C-FIBERS PLAY A ROLE BY ELICITING NEUROGENIC PAIN, INSULIN RESISTANCE IN DIABETES MELLITUS OR AGING, INHIBIT INSULIN ANTAGONIZING PEPTIDE, NOVO NORDISK A/S (DK) 2001-05-29 US disclosed
US-6166009-A N-substituted azaheterocyclic carboxylic acids and esters thereof NOVO NORDISK A/S (DK) 2000-12-26 US disclosed
US-6110913-A ANTIINFLAMMATORY AGENTS, ANALGESICS NOVO NORDISK A/S (DK) 2000-08-29 US disclosed
US-6071901-A TREATING PAIN, HYPERALGESIA AND/OR INFLAMMATORY CONDITIONS IN WHICH C-FIBERS PLAY A PATHOPHYSIOLOGICAL ROLE; INHIBITION OF NEUROGENIC INFLAMMATION INVOLVING THE RELEASE OF NEURO-PEPTIDE FROM PERIPHERAL AND CENTRAL ENDINGS OF SENSORY NERVES NOVO NORDISK A/S (DK) 2000-06-06 US disclosed
US-5874428-A A DRUG TREATING DIABETIC NEUROPATHY, MIGRAINE, NEUROGENIC INFLAMMATION OR RHEUMATOID ARTHRITIS NOVO NORDISK ALS (DK) 1999-02-23 US disclosed
EP-0820451-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1998-01-28 EP disclosed
WO-1996031498-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250326732-A1 CHROMEN-2-ONE MODULATORS OF POLRMT POLRMT, TFAM, POLM SLC6A2 4048/4885SLC6A3 4538/4885SLC6A4 4127/4885
US-20120130076-A1 Synthetic Multimerizing Agents FKBP1B, FKBP2, FKBP14 SLC6A2 4347/4885SLC6A3 4806/4885SLC6A4 4058/4885
US-20110152234-A1 Novel Compounds CNR1, ABCG2, CNR2 SLC6A2 2320/4885SLC6A3 1646/4885SLC6A4 2060/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.