SCHEMBL19302914

SCHEMBL19302914

Nc1ncnc2c1ncn2[C@@H]1O[C@H](CNS(=O)(=O)/C=C/CCC(=O)c2ccccc2-c2c(O)c(=O)c2=O)[C@@H](O)[C@H]1O

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPM2 O94759 1/20 0.51
IMPDH2 P12268 2/20 0.49
IMPDH1 P20839 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19302682 0.88 IMPDH2 (0.53) TRPM2IMPDH2IMPDH1
SCHEMBL19302703 0.88 IMPDH2 (0.51) TRPM2IMPDH2IMPDH1
SCHEMBL19302912 0.87 IMPDH2 (0.48) TRPM2IMPDH2IMPDH1
SCHEMBL19302909 0.86 HINT1 (0.56) TRPM2
SCHEMBL19302841 0.86 TRPM2 (0.53) TRPM2
SCHEMBL19302910 0.86 IMPDH2 (0.47) TRPM2IMPDH2IMPDH1
SCHEMBL19302911 0.85
SCHEMBL19302968 0.83 IMPDH2 (0.48) TRPM2IMPDH2IMPDH1
SCHEMBL19302871 0.81 GNMT (0.59)
SCHEMBL19302777 0.81 TRPM2 (0.52) TRPM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017059411-A9 INHIBITORS OF MENAQUINONE BIOSYNTHESIS MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2017-08-31 WO disclosed