SCHEMBL19331685

SCHEMBL19331685

O=C(O)CNC(=O)CCC/C=C\CCCCCCC/C=C\CCCCO

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 6/20 0.64
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
ALDH1A1 P00352 3/20 0.64
BLM P54132 2/20 0.64
KDM4E B2RXH2 1/20 0.64
USP2 O75604 1/20 0.64
POLB P06746 1/20 0.64
CYP3A4 P08684 1/20 0.64
MAPT P10636 1/20 0.64
HPGD P15428 1/20 0.64
ALOX15 P16050 1/20 0.64
APEX1 P27695 1/20 0.64
RECQL P46063 1/20 0.64
PMP22 Q01453 1/20 0.64
GPR18 Q14330 1/20 0.64
HSD17B10 Q99714 1/20 0.64
TDP1 Q9NUW8 1/20 0.64
SLC6A5 Q9Y345 1/20 0.64
PTPN1 P18031 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL413821 1.00 FAAH (0.64) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL19331672 0.96 MEN1 (0.67) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL12189673 0.87 PTPN1 (0.71) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL22717109 0.87 PTPN1 (0.71) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL13189678 0.85 PTPN1 (0.68) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL1424411 0.84 FAAH (0.88) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL1424413 0.84 FAAH (0.88) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL19331609 0.84 FAAH (0.62) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL20398921 0.84 FAAH (0.88) FAAHMEN1KMT2AALDH1A1BLM
SCHEMBL25764050 0.84 FAAH (0.88) FAAHMEN1KMT2AALDH1A1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240041831-A1 20-HETE RECEPTOR (GPR75) ANTAGONISTS AND METHODS OF USE NEW YORK MEDICAL COLLEGE 2024-02-08 US disclosed
US-11690825-B2 20-HETE receptor (GPR75) antagonists and methods of use BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-07-04 US disclosed
US-11690825-B2 20-HETE receptor (GPR75) antagonists and methods of use BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-07-04 US disclosed
US-11690825-B2 20-HETE receptor (GPR75) antagonists and methods of use BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-07-04 US disclosed
US-20200030291-A1 20-HETE RECEPTOR (GPR75) ANTAGONISTS AND METHODS OF USE NEW YORK MEDICAL COLLEGE 2020-01-30 US disclosed
US-20200030291-A1 20-HETE RECEPTOR (GPR75) ANTAGONISTS AND METHODS OF USE NEW YORK MEDICAL COLLEGE 2020-01-30 US disclosed
WO-2017156164-A1 20-HETE RECEPTOR (GPR75) ANTAGONISTS AND METHODS OF USE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-09-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240041831-A1 20-HETE RECEPTOR (GPR75) ANTAGONISTS AND METHODS OF USE GPR55, GPR65, GPR35 FAAH 352/4885MEN1 3401/4885KMT2A 3465/4885
US-20200030291-A1 20-HETE RECEPTOR (GPR75) ANTAGONISTS AND METHODS OF USE GPR55, GPR65, GPR35 FAAH 352/4885MEN1 3401/4885KMT2A 3465/4885
US-11690825-B2 20-HETE receptor (GPR75) antagonists and methods of use GPR55, GPR65, GPR35 FAAH 352/4885MEN1 3401/4885KMT2A 3465/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.