SCHEMBL19337640

SCHEMBL19337640

CC(=O)Nc1cccc(NC(=O)c2ccc(-c3ccccc3)cc2)c1C

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.72
RAB9A P51151 2/20 0.72
DHODH Q02127 1/20 0.59
MEN1 O00255 4/20 0.58
KMT2A Q03164 4/20 0.58
MAPT P10636 2/20 0.58
HPGD P15428 2/20 0.58
LMNA P02545 2/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HDAC1 Q13547 3/20 0.58
PDCD1 Q15116 1/20 0.56
CD274 Q9NZQ7 1/20 0.56
GRM5 P41594 1/20 0.54
POLB P06746 2/20 0.53
PTPN1 P18031 1/20 0.51
CACNA1B Q00975 1/20 0.51
APBA1 Q02410 1/20 0.51
KDM4E B2RXH2 1/20 0.51
APOBEC3A P31941 1/20 0.51
GFER P55789 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16330055 0.84 POLB (0.72) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL15290422 0.81 HPGD (0.80) NPC1RAB9ADHODHMEN1KMT2A
SCHEMBL14817806 0.80 ALDH1A1 (0.65) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL13053955 0.78 NPC1 (0.62) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL10212149 0.78 NPC1 (0.62) NPC1RAB9ADHODHMEN1KMT2A
SCHEMBL29788136 0.78 KDM4E (0.55) NPC1RAB9AHPGDLMNASMN1; SMN2
SCHEMBL2040639 0.76 FFAR2 (0.51) NPC1RAB9ADHODHMEN1KMT2A
SCHEMBL29788091 0.76 FFAR2 (0.51) NPC1RAB9ADHODHMEN1KMT2A
SCHEMBL11769542 0.76 POLB (0.77) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL30288146 0.76 POLB (0.77) NPC1RAB9AMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2291352-B1 N-ACYLTHIOUREA AND N-ACYLUREA INHIBITORS OF THE HEDGEHOG PROTEIN SIGNALLING PATHWAY CENTRE NAT RECH SCIENT (FR) 2017-09-13 EP disclosed