SCHEMBL1934698

SCHEMBL1934698

O=C(O)NCCN1CCCCC1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.61
CA1 P00915 3/20 0.61
CA2 P00918 3/20 0.61
CA9 Q16790 3/20 0.61
ALDH1A1 P00352 4/20 0.57
KDM4E B2RXH2 2/20 0.57
NPC1 O15118 1/20 0.56
POLB P06746 2/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
CYP1A2 P05177 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
RAB9A P51151 1/20 0.50
MAPK1 P28482 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL165673 0.98 CA12 (0.60) CA12CA1CA2CA9ALDH1A1
SCHEMBL21065340 0.89 CA12 (0.48) CA12CA1CA2CA9ALDH1A1
SCHEMBL9990508 0.88 SMN1; SMN2 (0.57) CA12CA1CA2CA9ALDH1A1
Cyclohexanol SCHEMBL9499967 0.88 CA12 (0.50) CA12CA1CA2CA9ALDH1A1
Cyclohexanol SCHEMBL9497715 0.88 CA12 (0.50) CA12CA1CA2CA9ALDH1A1
SCHEMBL7068538 0.86 RAD52 (0.55) CA12CA1CA2CA9ALDH1A1
SCHEMBL9990414 0.85 SMN1; SMN2 (0.53) CA12CA1CA2CA9ALDH1A1
SCHEMBL3893911 0.84 CA12 (0.63) CA12CA1CA2CA9ALDH1A1
SCHEMBL2755862 0.83 RAD52 (0.53) CA12CA1CA2CA9ALDH1A1
SCHEMBL18824247 0.83 HDAC2 (0.49) CA12CA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614211-B2 Certain chemical entities, compositions, and methods NEUPHARMA, INC. (US) 2013-12-24 US claimed
US-20130040945-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA, INC. 2013-02-14 US claimed
WO-2013023145-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS NEUPHARMA, INC. (US) 2013-02-14 WO claimed
WO-2024019936-A1 NANOMATERIALS COMPRISING TRIOLS BEAM THERAPEUTICS INC. (US) 2024-01-25 WO disclosed
US-20230331737-A1 MTORC1 MODULATORS AND USES THEREOF AEOVIAN PHARMACEUTICALS, INC. 2023-10-19 US disclosed
US-20230151052-A1 NEUROSTEROID COMPOUNDS AND METHODS FOR THEIR PREPARATION AND USE IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS THE TEXAS A&M UNIVERSITY SYSTEM 2023-05-18 US disclosed
US-11542296-B2 Neurosteroid compounds and methods for their preparation and use in treating central nervous system disorders THE TEXAS A&M UNIVERSITY SYSTEM (US) 2023-01-03 US disclosed
EP-3950692-A1 NOVEL TRICYCLIC COMPOUNDS AbbVie Inc. (US) 2022-02-09 EP disclosed
US-20210238220-A1 NEUROSTEROID COMPOUNDS AND METHODS FOR THEIR PREPARATION AND USE IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2021-08-05 US disclosed
CN-109053742-B Novel tricyclic compounds ABBVIE 公司 2021-06-15 CN disclosed
US-20210061813-A1 NOVEL TRICYCLIC COMPOUNDS ABBVIE INC. (US) 2021-03-04 US disclosed
CN-102498095-A Indoline derivatives TOKYO INST TECH 2012-06-13 CN disclosed
US-20110311474-A1 Novel Tricyclic Compounds ABBOTT LABORATORIES (US) 2011-12-22 US disclosed
WO-2011068881-A1 NOVEL TRICYCLIC COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-09 WO disclosed
US-7671072-B2 Aminopyrazole derivatives as GSK-3 inhibitors PFIZER INC. (US) 2010-03-02 US disclosed
WO-2009033165-A1 HYPOXIA ACTIVATED PRODRUGS OF BIS-ALKYLATING AGENTS THRESHOLD PHARMACEUTICALS, INC. (US) 2009-03-12 WO disclosed
US-20070276010-A1 Aminopyrazole Derivatives as Gsk-3 Inhibitors BENBOW JOHN W 2007-11-29 US disclosed
US-6740741-B2 SUCH AS (2-(1-PIPERIDINE)ETHYL)CARBAMATE FOR THE DEACIDIFICATION OF PAPER MATERIAL CONSIGLIO NAZIONALE DELLE RICERCHE (IT) 2004-05-25 US disclosed
US-20030065153-A1 Novel diazo derivatives and process for their preparation ZAPPALA ANTONIO (IT) 2003-04-03 US disclosed
EP-1273568-A2 Novel diazo derivatives and process for their preparation CONSIGLIO NAZIONALE DELLE RICERCHE (IT) 2003-01-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230151052-A1 NEUROSTEROID COMPOUNDS AND METHODS FOR THEIR PREPARATION AND USE IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS CYP11B2, CYP21A2, CYP11B1 CA12 2607/4885CA1 1841/4885CA2 3374/4885
US-20070276010-A1 Aminopyrazole Derivatives as Gsk-3 Inhibitors GSK3B, GSK3A, GSKIP CA12 3894/4885CA1 2361/4885CA2 3175/4885
US-20210238220-A1 NEUROSTEROID COMPOUNDS AND METHODS FOR THEIR PREPARATION AND USE IN TREATING CENTRAL NERVOUS SYSTEM DISORDERS CYP11B2, CYP21A2, CYP11B1 CA12 2607/4885CA1 1841/4885CA2 3374/4885
US-20030065153-A1 Novel diazo derivatives and process for their preparation DDT, DDC, ACMSD CA12 1321/4885CA1 1594/4885CA2 2144/4885
US-20230331737-A1 MTORC1 MODULATORS AND USES THEREOF MTOR, RPTOR, RICTOR CA12 4798/4885CA1 4771/4885CA2 4043/4885
US-20210061813-A1 NOVEL TRICYCLIC COMPOUNDS CYP11B2, CYP11B1, ABCB1 CA12 641/4885CA1 1857/4885CA2 1833/4885
US-11542296-B2 Neurosteroid compounds and methods for their preparation and use in treating central nervous system disorders CYP11B2, CYP21A2, CYP11B1 CA12 2607/4885CA1 1841/4885CA2 3374/4885
US-20110311474-A1 Novel Tricyclic Compounds CYP11B2, CYP11B1, ABCB1 CA12 641/4885CA1 1857/4885CA2 1833/4885
US-20130040945-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS RXRG, ARNT, RARS2 CA12 986/4885CA1 2686/4885CA2 2121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.