SCHEMBL193474

SCHEMBL193474

CC(C)(C)OC(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)O

nearest known ligand 0.73

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.73
ITGB3 P05106 3/20 0.67
ITGA2B P08514 3/20 0.67
BCL2 P10415 1/20 0.67
PPARG P37231 3/20 0.65
ACE P12821 2/20 0.65
PPARA Q07869 2/20 0.63
YAP1 P46937 1/20 0.62
MME P08473 1/20 0.61
CPA1 P15085 1/20 0.61
ACE2 Q9BYF1 1/20 0.61
GPR34 Q9UPC5 2/20 0.60
HDAC8 Q9BY41 1/20 0.59
CTSS P25774 2/20 0.58
CTSL P07711 1/20 0.58
CTSB P07858 1/20 0.58
CTSK P43235 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL193473 1.00 PTPN1 (0.73) PTPN1ITGB3ITGA2BBCL2PPARG
SCHEMBL2891538 1.00 PTPN1 (0.73) PTPN1ITGB3ITGA2BBCL2PPARG
SCHEMBL28267499 0.95 PTPN1 (0.77) PTPN1ITGB3ITGA2BBCL2PPARG
SCHEMBL28267496 0.95 PTPN1 (0.77) PTPN1ITGB3ITGA2BBCL2PPARG
SCHEMBL464744 0.93 PTPN1 (0.65) PTPN1ITGB3ITGA2BBCL2PPARG
Phenylalanine Methyl Ester SCHEMBL28119144 0.91 PTPN1 (0.63) PTPN1ITGB3ITGA2BBCL2PPARG
SCHEMBL3350988 0.91 BCL2 (0.64) PTPN1ITGB3ITGA2BBCL2PPARG
SCHEMBL9752771 0.91 BCL2 (0.64) PTPN1ITGB3ITGA2BBCL2PPARG
SCHEMBL9752770 0.91 BCL2 (0.64) PTPN1ITGB3ITGA2BBCL2PPARG
SCHEMBL3500186 0.91 BCL2 (0.64) PTPN1ITGB3ITGA2BBCL2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 166 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106188231-B Synthesis and application of pasireotide pentapeptide intermediate 中国医学科学院药物研究所 2021-10-22 CN claimed
CN-106188231-A The synthesis of pasireotide pentapeptide intermediate and application 中国医学科学院药物研究所 2016-12-07 CN claimed
US-12625431-B2 EUV resist underlayer film-forming composition NISSAN CHEMICAL CORPORATION (JP) 2026-05-12 US disclosed
US-20260015313-A1 AMINO ACID ACTIVE ESTER AND SALT THEREOF PEPTIDREAM INC (JP) 2026-01-15 US disclosed
EP-4534524-A1 AMINO ACID ACTIVE ESTER AND SALT THEREOF PeptiDream Inc. (JP) 2025-04-09 EP disclosed
US-20240122951-A1 METHOD TO TREAT LIPID DYSREGULATION BY MODULATING ACTIVITY OF PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9 (PCSK9) PROTEIN WITH SMALL MOLECULE LIGANDS SRX CARDIO, LLC 2024-04-18 US disclosed
US-11834406-B2 Conjugates of cell binding molecules with cytotoxic agents HANGZHOU DAC BIOTECH CO., LTD. (CN) 2023-12-05 US disclosed
US-11771710-B2 Method to treat lipid dysregulation by modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9) protein activity with small molecule ligands SRX CARDIO, LLC (US) 2023-10-03 US disclosed
US-11767294-B2 Conjugates of cell binding molecules with cytotoxic agents HANGZHOU DAC BIOTECH CO., LTD. (CN) 2023-09-26 US disclosed
CN-116143678-A Conjugate linker, cell-binding molecule-drug conjugate containing the same, and preparation and application thereof 杭州多禧生物科技有限公司 2023-05-23 CN disclosed
CN-110099682-B Coupled connector, cell binding molecule-drug conjugate containing same, and preparation and application thereof 杭州多禧生物科技有限公司 2023-03-31 CN disclosed
EP-0195667-A2 Cardiotonic quinazoline derivatives KYOWA HAKKO KOGYO KABUSHIKI KAISHA (JP) 1986-09-24 EP disclosed
EP-0190588-A1 Quinazolino-1,4-benzodiazepin-6,9-diones, processes for their preparation and pharmaceutical compositions containing them MERCK & CO. INC. (US) 1986-08-13 EP disclosed
US-4554272-A CHOLECYSTOKININ INHIBITORS MERCK & CO., INC. (US) 1985-11-19 US disclosed
US-4535169-A 5H-6-oxo-2,3,4,4a,7,7a-hexahydropyrano[2,3-b]pyrrole and the preparation thereof THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1985-08-13 US disclosed
US-4407746-A Cyclohexyl and phenyl substituted enkephalins G. D. SEARLE & CO. (US) 1983-10-04 US disclosed
US-4301045-A RESIN PEPTIDES ARMOUR PHARMACEUTICAL COMPANY (US) 1981-11-17 US disclosed
US-4146614-A TREATMENT OF SCHIZOPHRENIA STATE OF MICHIGAN (US) 1979-03-27 US disclosed
US-3974135-A Synthetic decapeptide having the activity of the luteinizing hormone releasing hormone and method for producing the same FOLKERS KARL 1976-08-10 US disclosed
US-3953416-A Synthetic decapeptide having the activity of the luteinizing hormone releasing hormone and method for manufacturing the same FOLKERS KARL 1976-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260015313-A1 AMINO ACID ACTIVE ESTER AND SALT THEREOF NSUN3, BCAT1, SLC43A1 PTPN1 827/4885ITGB3 2864/4885ITGA2B 3805/4885
US-11767294-B2 Conjugates of cell binding molecules with cytotoxic agents CD4, CD2, CD47 PTPN1 1021/4885ITGB3 314/4885ITGA2B 442/4885
US-12625431-B2 EUV resist underlayer film-forming composition EEF1A1, ARF1, EMG1 PTPN1 912/4885ITGB3 358/4885ITGA2B 496/4885
US-20240122951-A1 METHOD TO TREAT LIPID DYSREGULATION BY MODULATING ACTIVITY OF PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9 (PCSK9) PROTEIN WITH SMALL MOLECULE LIGANDS PCSK9, LDLR, PCSK7 PTPN1 779/4885ITGB3 3292/4885ITGA2B 3936/4885
US-11771710-B2 Method to treat lipid dysregulation by modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9) protein activity with small molecule ligands PCSK9, LDLR, PCSK7 PTPN1 786/4885ITGB3 3310/4885ITGA2B 3985/4885
US-11834406-B2 Conjugates of cell binding molecules with cytotoxic agents CD4, CD2, CD47 PTPN1 1161/4885ITGB3 269/4885ITGA2B 426/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.