SCHEMBL19359258

SCHEMBL19359258

Cc1ccn(-c2cccc(B(O)O)n2)c1C

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
ATM Q13315 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CDC7 O00311 1/20 0.31
CDK2 P24941 1/20 0.31
ROCK1 Q13464 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2559276 0.76 KDR (0.42)
SCHEMBL18586553 0.73 ALDH1A1 (0.35) NPC1MAPTRAB9AATMSMN1; SMN2
SCHEMBL2563617 0.71 RAB9A (0.69) NPC1MAPTRAB9AATMSMN1; SMN2
SCHEMBL29956895 0.71 HRH4 (0.38)
SCHEMBL2556317 0.70 PIK3CA (0.35) MAPTL3MBTL1CDC7CDK2ROCK1
SCHEMBL20067383 0.67 ENPP2 (0.36)
SCHEMBL15330702 0.67 ALDH1A1 (0.41) NPC1MAPTRAB9AATMSMN1; SMN2
SCHEMBL956317 0.67 CCR1 (0.48) NPC1RAB9ASMN1; SMN2
SCHEMBL29955389 0.67 CCR1 (0.48) NPC1RAB9ASMN1; SMN2
SCHEMBL15845752 0.66 HSD11B1 (0.42) MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017161145-A1 TRIAZOLOPYRIDINE INHIBITORS OF MYELOPEROXIDASE AND/OR EPX BRISTOL-MYERS SQUIBB COMPANY (US) 2017-09-21 WO disclosed