SCHEMBL19360397

SCHEMBL19360397

CCn1c(Cc2ccc(C(F)(F)F)nc2)cc2cc(C(=O)OC)ccc21

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORC P51449 12/20 0.51
KDM4E B2RXH2 1/20 0.45
NR1H4 Q96RI1 1/20 0.43
ACSS2 Q9NR19 1/20 0.39
CNR2 P34972 1/20 0.39
CSF1R P07333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19360401 0.89 RORC (0.51) RORC
SCHEMBL19360388 0.85 RORC (0.55) RORCKDM4EACSS2CNR2
SCHEMBL19360394 0.82 RORC (0.64) RORC
SCHEMBL19360605 0.82 IDH1 (0.47) RORCKDM4ENR1H4ACSS2CNR2
SCHEMBL19360520 0.78 KIF11 (0.51) RORCKDM4EACSS2
SCHEMBL18440914 0.76 RORC (0.52) RORCKDM4E
SCHEMBL19360593 0.75 KDM4E (0.43) RORCKDM4EACSS2
SCHEMBL20634743 0.75 RORC (0.46) RORCKDM4ECNR2
SCHEMBL19360398 0.75 HTT (0.45) RORCKDM4ENR1H4
SCHEMBL18440701 0.73 RORC (0.55) RORCACSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107531679-B Aromatic amide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-02 CN disclosed
CN-107531679-A Aromatic amides analog derivative, its preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2018-01-02 CN disclosed
WO-2017157332-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATIONS THEREOF 江苏恒瑞医药股份有限公司 2017-09-21 WO disclosed