SCHEMBL19405232

SCHEMBL19405232

C=C(C)C(=O)c1ccc(CN)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.57
THRB P10828 1/20 0.57
LOXL2 Q9Y4K0 4/20 0.53
MAPT P10636 1/20 0.53
HDAC3 O15379 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
KDM4E B2RXH2 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
F10 P00742 1/20 0.45
NOS3 P29474 2/20 0.42
NOS1 P29475 2/20 0.42
NOS2 P35228 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
ABAT P80404 1/20 0.41
TPSAB1 Q15661 3/20 0.41
HRH3 Q9Y5N1 1/20 0.39
PSIP1 O75475 1/20 0.38
SMYD3 Q9H7B4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28670034 0.82 MAPT (0.71) THRATHRBMAPTSMN1; SMN2KMT2A
SCHEMBL11839721 0.82 LOXL2 (0.58) THRATHRBLOXL2MAPTSMN1; SMN2
SCHEMBL9850596 0.82 THRA (0.64) THRATHRBMAPTSMN1; SMN2KMT2A
SCHEMBL21840691 0.82 THRA (0.59) THRATHRBMAPTSMN1; SMN2NOS3
SCHEMBL18286692 0.80 THRB (0.57) THRATHRBMAPTHDAC6KMT2A
Ethylene SCHEMBL11090983 0.79 KMT2A (0.61) LOXL2MAPTHDAC3HDAC6NCOR2
SCHEMBL7493555 0.79 HDAC3 (0.57) LOXL2HDAC3HDAC6NCOR2KDM4E
SCHEMBL2399333 0.79 LOXL2 (0.52) LOXL2HDAC3HDAC6NCOR2KDM4E
SCHEMBL856509 0.79 KMT2A (0.67) LOXL2MAPTHDAC3HDAC6NCOR2
SCHEMBL11645482 0.78 THRB (0.75) THRATHRBMAPTKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017163264-A1 BLOCKING TOLL-LIKE RECEPTOR 9 SIGNALING WITH SMALL MOLECULE ANTAGONIST COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2017-09-28 WO disclosed