SCHEMBL19413239

SCHEMBL19413239

CCCCCCC(C)(CCCCCC)C(=O)NCc1nnc(C)[nH]1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 4/20 0.33
CCR2 P41597 2/20 0.32
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CXCR4 P61073 1/20 0.32
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
MAPT P10636 2/20 0.32
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
ACAT1 P24752 1/20 0.32
SOAT1 P35610 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31
CES2 O00748 1/20 0.30
LPAR1 Q92633 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20625833 0.89 CCR2 (0.39) EPHX1CCR2CCR1CCR5CXCR4
SCHEMBL20363209 0.72 FAAH (0.48) EPHX1CES2
SCHEMBL20625835 0.71 HRH3 (0.44)
SCHEMBL20363242 0.71 FAAH (0.47) EPHX1CES2
SCHEMBL20363294 0.70 RAB9A (0.49) MAPTKDM4EALOX15TSHR
SCHEMBL20363296 0.69 RAB9A (0.51) GAAMAPTKDM4EALOX15TSHR
SCHEMBL19413256 0.69 S1PR1 (0.33) EPHX1CCR2CCR1CCR5CXCR4
SCHEMBL20363229 0.69 RAB9A (0.50) GAAMAPTKDM4EALOX15TSHR
SCHEMBL23502458 0.68 PLA2G2A (0.50) ALOX15TSHRMEN1KMT2A
SCHEMBL18743801 0.68 EPHX1 (0.41) EPHX1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9776996-B2 Substituted 6,5-fused bicyclic heteroaryl compounds Epizyme, Inc. (US) 2017-10-03 US disclosed