SCHEMBL19418286

SCHEMBL19418286

CC1COc2cc(F)ccc2N1N

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 6/20 0.44
NR3C1 P04150 4/20 0.44
PGR P06401 1/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HCRTR2 O43614 1/20 0.39
CA2 P00918 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
TSHR P16473 1/20 0.38
ROCK1 Q13464 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
AKR1B1 P15121 1/20 0.35
ALDH1A1 P00352 1/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
LTA4H P09960 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25883473 0.82 NR3C1 (0.45) NR3C2NR3C1PGRMEN1KMT2A
SCHEMBL9029862 0.76 NR3C2 (0.56) NR3C2NR3C1PGRMEN1KMT2A
SCHEMBL9029850 0.76 NR3C2 (0.56) NR3C2NR3C1PGRMEN1KMT2A
SCHEMBL19030251 0.73 DRD2 (0.47) NR3C2NR3C1PGRMEN1KMT2A
SCHEMBL20804963 0.69 NR3C2 (0.52) NR3C2NR3C1PGRMEN1KMT2A
SCHEMBL19418129 0.68 ALDH1A1 (0.43) NR3C2NR3C1L3MBTL1KDM4EHTT
Diethylamine SCHEMBL9700231 0.68 SMN1; SMN2 (0.45) MEN1KMT2ACA2L3MBTL1ALDH1A1
SCHEMBL3485497 0.67 NR3C2 (0.38) NR3C2NR3C1PGRCA2DRD2
SCHEMBL30457404 0.67 ADRA2A (0.39) HCRTR2CA2AKR1B1
SCHEMBL25723206 0.67 ADRA2A (0.39) HCRTR2CA2AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925757-B1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES NOVARTIS AG (CH) 2017-10-04 EP disclosed