SCHEMBL19457426

SCHEMBL19457426

C=C(N)c1ccc(Cc2ccc(C(=C)N)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.50
PLA2G2A P14555 1/20 0.50
KMT2A Q03164 1/20 0.46
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
ALDH1A1 P00352 2/20 0.43
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CYP17A1 P05093 1/20 0.42
LMNA P02545 1/20 0.40
PRSS1 P07477 2/20 0.39
PRSS2 P07478 2/20 0.39
PRSS3 P35030 2/20 0.39
F10 P00742 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
SLC22A2 O15244 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10092625 0.93 CYP17A1 (0.52) PLA2G10PLA2G2AKMT2AADRA2AADRA2B
SCHEMBL15893699 0.82 LOXL2 (0.60) F10LOXL2HDAC6
SCHEMBL13362346 0.82 PRSS1 (0.60) PLA2G10PLA2G2ATSHRPRSS1PRSS2
SCHEMBL14565742 0.80 SMN1; SMN2 (0.61) ALDH1A1TDP1PRSS1SMN1; SMN2CA2
SCHEMBL22872694 0.80 NOS1 (0.52) KMT2AALDH1A1CYP3A4LMNALOXL2
SCHEMBL451895 0.77 PLA2G10 (0.53) PLA2G10PLA2G2AKMT2AADRA2AADRA2B
SCHEMBL20117499 0.77 THRB (0.53) KMT2AALDH1A1ESR1ESR2SMN1; SMN2
SCHEMBL18726920 0.75 PLA2G10 (0.33) PLA2G10PLA2G2ACYP17A1
SCHEMBL8178806 0.75 CYP2C9 (0.37) KMT2AALDH1A1PRSS1PRSS2PRSS3
SCHEMBL7134591 0.74 PLA2G10 (0.83) PLA2G10PLA2G2AKMT2AALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017174879-A1 COMPOUNDS FOR USE IN THE TREATMENT OF CANCER UNIVERSITY OF OULU (FI) 2017-10-12 WO disclosed