SCHEMBL1948375

SCHEMBL1948375

COCC(=O)N1CCc2ccc(NCc3ccc(Cl)cc3)cc21

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.51
DRD4 P21917 8/20 0.51
NOTUM Q6P988 1/20 0.46
HSD17B3 P37058 1/20 0.43
MEN1 O00255 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
KMT2A Q03164 1/20 0.43
PTPN11 Q06124 1/20 0.43
XIAP P98170 1/20 0.42
BIRC2 Q13490 1/20 0.42
THRB P10828 1/20 0.42
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1950469 0.91 DRD4 (0.50) DRD2DRD4NOTUMPTPN11THRB
SCHEMBL1950711 0.91 DRD2 (0.48) DRD2DRD4NOTUMHSD17B3MEN1
SCHEMBL1950239 0.86 NOTUM (0.64) DRD2DRD4NOTUMHSD17B3KMT2A
SCHEMBL2641013 0.86 PTPN11 (0.41) DRD2DRD4HSD17B3MEN1ADRA1D
SCHEMBL1948851 0.83 NOTUM (0.44) DRD2DRD4NOTUMHSD17B3THRB
SCHEMBL1950866 0.82 DRD2 (0.48) DRD2DRD4NOTUMMEN1KMT2A
SCHEMBL1950717 0.82 KMT2A (0.49) HSD17B3MEN1KMT2AMAPTLMNA
SCHEMBL2641060 0.80 LMNA (0.44) DRD2DRD4NOTUMHSD17B3THRB
SCHEMBL20536797 0.78 MAPT (0.61) THRBMAPTLMNAPOLB
SCHEMBL1948510 0.77 NOTUM (0.64) DRD2DRD4NOTUMHSD17B3THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438055-B1 DIHYDROINDOLE AND TETRAHYDROISOQUINOLINE DERIVATIVES USEFUL AS POTASSIUM CHANNEL INHIBITORS JAPAN TOBACCO INC (JP) 2018-10-24 EP claimed
US-8426442-B2 Compounds XENTION LTD (GB) 2013-04-23 US claimed
EP-2438055-B1 DIHYDROINDOLE AND TETRAHYDROISOQUINOLINE DERIVATIVES USEFUL AS POTASSIUM CHANNEL INHIBITORS JAPAN TOBACCO INC (JP) 2018-10-24 EP disclosed
US-8426442-B2 Compounds XENTION LTD (GB) 2013-04-23 US disclosed
US-20110136860-A1 Compounds XENTION LTD. (GB) 2011-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110136860-A1 Compounds NR3C2, NR5A1, NR0B2 DRD2 385/4885DRD4 739/4885NOTUM 2101/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.