Fumaric Acid

Fumaric Acid

SCHEMBL194895

CCCCCCCCOC(=O)[C@@H]1C[C@@H]2CCC[C@@H]2N1C(=O)[C@H](C)N[C@@H](CCc1ccccc1)C(=O)OCC.O=C(O)/C=C/C(=O)O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB1ADRB2ATP4AATP4BAXLCHRM2CHRM3DRD2FLT3HRH1HTR2AHTR2BHTR2CKCNH2KMT2AMAP2K1MAP2K2MEN1MLNRPLK4RENS1PR1SLC6A2SLC6A4atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 2/20 0.72
KMT2A known ✓ Q03164 2/20 0.72
ACE P12821 14/20 0.72
CYP3A4 P08684 1/20 0.72
ALOX15 P16050 1/20 0.72
LMNA P02545 2/20 0.69
USP2 O75604 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.58
ABCB11 O95342 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL9773179 1.00 ACE (0.72) ACEMEN1KMT2ACYP3A4ALOX15
Maleic Acid SCHEMBL9773162 1.00 ACE (0.72) ACEMEN1KMT2ACYP3A4ALOX15
Maleic Acid SCHEMBL9773197 0.97 ACE (0.69) ACEMEN1KMT2ACYP3A4ALOX15
SCHEMBL9775445 0.96 ACE (0.77) ACEMEN1KMT2ACYP3A4ALOX15
SCHEMBL9773138 0.96 ACE (0.77) ACEMEN1KMT2ACYP3A4ALOX15
SCHEMBL9593609 0.96 ACE (0.77) ACEMEN1KMT2ACYP3A4ALOX15
SCHEMBL9775474 0.96 ACE (0.77) ACEMEN1KMT2ACYP3A4ALOX15
SCHEMBL9773238 0.96 ACE (0.77) ACEMEN1KMT2ACYP3A4ALOX15
SCHEMBL9773120 0.96 ACE (0.77) ACEMEN1KMT2ACYP3A4ALOX15
SCHEMBL9773161 0.96 ACE (0.77) ACEMEN1KMT2ACYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240002935-A1 GENETIC METHOD FOR DIAGNOSIS AND TREATMENT OF PRE AND POST CORONAVIRUS INFECTIONS GENETICURE INC. 2024-01-04 US claimed
EP-4132653-A1 GENETIC METHOD FOR DIAGNOSIS AND TREATMENT OF PRE AND POST CORONAVIRUS INFECTIONS Geneticure Inc. (US) 2023-02-15 EP claimed
US-12453717-B1 Methods of treating symptoms of coronavirus infection with viral protease inhibitors Accencio LC (US) 2025-10-28 US disclosed
US-12083099-B2 Methods of treating symptoms of coronavirus infection with viral protease inhibitors Accencio LLC (US) 2024-09-10 US disclosed
US-20240002935-A1 GENETIC METHOD FOR DIAGNOSIS AND TREATMENT OF PRE AND POST CORONAVIRUS INFECTIONS GENETICURE INC. 2024-01-04 US disclosed
US-11761043-B2 Machine assay and analysis for selecting antihypertensive drugs GENETICURE INC. (US) 2023-09-19 US disclosed
US-11674179-B2 Therapeutic regimen for hypertension GENETICURE INC. (US) 2023-06-13 US disclosed
US-20230113114-A1 METHODS OF TREATING SYMPTOMS OF CORONAVIRUS INFECTION WITH VIRAL PROTEASE INHIBITORS Accencio LLC 2023-04-13 US disclosed
EP-4132653-A1 GENETIC METHOD FOR DIAGNOSIS AND TREATMENT OF PRE AND POST CORONAVIRUS INFECTIONS Geneticure Inc. (US) 2023-02-15 EP disclosed
US-20170129915-A1 THERAPEUTIC AGENT FOR DISEASES ASSOCIATED WITH NERVE AXON DYSFUNCTION, INCLUDING THERAPEUTIC AGENT FOR ALZHEIMER'S DISEASE RESILIO COMPANY LIMITED (JP) 2017-05-11 US disclosed
US-9453000-B2 Polycyclic compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2016-09-27 US disclosed
US-20110009619-A1 POLYCYCLIC COMPOUND EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-01-13 US disclosed
WO-2010098495-A1 IMIDAZOLYLPYRAZINE DERIVATIVES EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-09-02 WO disclosed
WO-2010098488-A1 ARYL IMIDAZOLE COMPOUNDS AND THEIR USE AS BETA AMYLOID PRODUCTION INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-09-02 WO disclosed
WO-2010098487-A1 NITROGEN-CONTAINING FUSED HETEROCYCLIC COMPOUNDS AND THEIR USE AS BETA AMYLOID PRODUCTION INHIBITORS EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-09-02 WO disclosed
US-20100130537-A1 CINNAMIDE COMPOUNDS FOR DEMENTIA EISAI R&D MANAGEMENT CO., LTD (JP) 2010-05-27 US disclosed
EP-2181992-A1 POLYCYCLIC COMPOUND Eisai R&D Management Co., Ltd. (JP) 2010-05-05 EP disclosed
EP-2148673-A1 CINNAMIDE COMPOUNDS FOR DEMENTIA Eisai R&D Management Co., Ltd. (JP) 2010-02-03 EP disclosed
US-20090062529-A1 MULTI-CYCLIC COMPOUNDS EISAI R&D MANAGEMENT CO., LTD., (JP) 2009-03-05 US disclosed
WO-2008139984-A1 CINNAMIDE COMPOUNDS FOR DEMENTIA EISAI R & D MANAGEMENT CO., LTD. (JP) 2008-11-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100130537-A1 CINNAMIDE COMPOUNDS FOR DEMENTIA GRIN1, GRIN2A, GRIN3A MEN1 1880/4885KMT2A 183/4885ACE 115/4885
US-12453717-B1 Methods of treating symptoms of coronavirus infection with viral protease inhibitors ACE, ACE2, TMPRSS2 MEN1 4436/4885KMT2A 708/4885ACE 1/4885
US-20110009619-A1 POLYCYCLIC COMPOUND APP, BACE1, PSEN1 MEN1 424/4885KMT2A 1666/4885ACE 325/4885
US-20170129915-A1 THERAPEUTIC AGENT FOR DISEASES ASSOCIATED WITH NERVE AXON DYSFUNCTION, INCLUDING THERAPEUTIC AGENT FOR ALZHEIMER'S DISEASE GAP43, NGF, BDNF MEN1 4095/4885KMT2A 4685/4885ACE 2747/4885
US-12083099-B2 Methods of treating symptoms of coronavirus infection with viral protease inhibitors ACE, ACE2, TMPRSS2 MEN1 3805/4885KMT2A 896/4885ACE 1/4885
US-20090062529-A1 MULTI-CYCLIC COMPOUNDS APP, BACE1, PSEN1 MEN1 531/4885KMT2A 2179/4885ACE 166/4885
US-20230113114-A1 METHODS OF TREATING SYMPTOMS OF CORONAVIRUS INFECTION WITH VIRAL PROTEASE INHIBITORS ACE, ACE2, TMPRSS2 MEN1 3805/4885KMT2A 896/4885ACE 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.