Chelerythrine

Chelerythrine

SCHEMBL195109

COc1ccc2c(c[n+](C)c3c4cc5c(cc4ccc23)OCO5)c1OC.[Cl-]

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBDKRB2CHRM1CHRM2CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNGGUCY1A1GUCY1A2GUCY1B1GUCY1B2NAMPTPTAFRSLC10A2SLC6A2SLC6A3TACR1dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Chelerythrine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 5/20 1.00
CHRM1 known ✓ P11229 2/20 0.50
ALDH1A1 P00352 7/20 1.00
MAPT P10636 7/20 1.00
SMN1; SMN2 Q16637 7/20 1.00
HPGD P15428 5/20 1.00
MAPK1 P28482 5/20 1.00
KMT2A Q03164 5/20 1.00
BCHE P06276 5/20 1.00
LMNA P02545 5/20 1.00
RAC1 P63000 4/20 1.00
GMNN O75496 2/20 1.00
POLB P06746 2/20 1.00
BLM P54132 2/20 1.00
PMP22 Q01453 2/20 1.00
NPSR1 Q6W5P4 2/20 1.00
BAD Q92934 2/20 1.00
PRKCE Q02156 1/20 1.00
CYP3A4 P08684 5/20 0.98
MEN1 O00255 4/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chelerythrine SCHEMBL30207103 1.00 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL29357531 0.99 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL30527168 0.99 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL30527167 0.99 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL288915 0.99 ALDH1A1 (1.00) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL4016265 0.98 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL4980861 0.98 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL288916 0.98 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL3319851 0.98 ALDH1A1 (0.98) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1
Chelerythrine SCHEMBL513051 0.95 ALDH1A1 (0.90) ALDH1A1MAPTSMN1; SMN2HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 792 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026090557-A1 SYSTEMS AND METHODS FOR PROCESSING ISM AND MCAS CLINICAL TRIAL DATA TELIOS PHARMA INC. (US) 2026-04-30 WO claimed
US-12472259-B2 PKC inhibitors for the treatment of septic cholestasis with polymethine dye targeting SMARTDYELIVERY GMBH (DE) 2025-11-18 US claimed
US-20250268913-A1 PKC INHIBITORS FOR THE TREATMENT OF SEPTIC CHOLESTASIS WITH CTM TARGETING SMARTDYELIVERY GMBH (DE) 2025-08-28 US claimed
US-20240082310-A1 BONE MARROW DERIVED NEUROKININ-1 RECEPTOR POSITIVE (NK1R+) MESENCHYMAL STEM CELLS FOR THERAPEUTIC APPLICATIONS BIOCARDIA INC (US) 2024-03-14 US claimed
US-20230025865-A1 COMPOSITIONS AND METHODS FOR SYSTEMIC DELIVERY OF Bcl-2 AND Bcl-xL ANTAGONISTS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2023-01-26 US claimed
CN-114786654-A Compositions and methods for systemic delivery of Bcl-2 and Bcl-xL antagonists 密执安大学评议会 2022-07-22 CN claimed
EP-3878947-A2 MATURATION OF MAMMALIAN HEPATOCYTES Takara Bio Europe AB (SE) 2021-09-15 EP claimed
US-20210189332-A1 MATURATION OF MAMMALIAN HEPATOCYTES TAKARA BIO EUROPE AB (SE) 2021-06-24 US claimed
WO-2021119439-A1 COMPOSITIONS AND METHODS FOR SYSTEMIC DELIVERY OF BCL-2 AND BCL-XL ANTAGONISTS THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2021-06-17 WO claimed
US-10913932-B2 Maturation of mammalian hepatocytes TAKARA BIO EUROPE AB (SE) 2021-02-09 US claimed
US-6407058-B1 Modifying the permeability of physiological barriers EISAI CO., LIMITED (JP) 2002-06-18 US claimed
JP-2001501618-A 2001-02-06 JP claimed
WO-1999041984-A9 INTERACTION BETWEEN THE MEC1-DEPENDENT DNA SYNTHESIS CHECKPOINT AND G1 CYCLIN FUNCTION IN $i(SACCAROMYCES CEREVISIAE) HUTCHINSON FRED CANCER RES (US) 1999-11-04 WO claimed
EP-0949917-A1 SUBSTANCES AND THEIR USES Eisai Co., Ltd. (JP) 1999-10-20 EP claimed
WO-1999041984-A1 INTERACTION BETWEEN THE MEC1-DEPENDENT DNA SYNTHESIS CHECKPOINT AND G1 CYCLIN FUNCTION IN $i(SACCAROMYCES CEREVISIAE) FRED HUTCHINSON CANCER RESEARCH CENTER (US) 1999-08-26 WO claimed
WO-1998014186-A1 SUBSTANCES AND THEIR USES EISAI CO., LIMITED (JP) 1998-04-09 WO claimed
WO-1997004761-A9 METHODS AND COMPOSITIONS FOR TREATING CELL PROLIFERATIVE DISORDERS 1997-05-29 WO claimed
WO-1997004761-A1 METHODS AND COMPOSITIONS FOR TREATING CELL PROLIFERATIVE DISORDERS TRUSTEES OF BOSTON UNIVERSITY (US) 1997-02-13 WO claimed
US-4683133-A PUMPING ALKALOID SALT SOLUTIONS ON GUMS VIPONT LABORATORIES, INC. (US) 1987-07-28 US claimed
US-4590061-A BENZO-C-PHENANTHRIDINE ALKALOIDS VIPONT LABORATORIES, INC. (US) 1986-05-20 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230025865-A1 COMPOSITIONS AND METHODS FOR SYSTEMIC DELIVERY OF Bcl-2 AND Bcl-xL ANTAGONISTS BCL2, BCL2L2, BCL2L1 ACHE 4546/4885CHRM1 4884/4885ALDH1A1 2779/4885
US-12472259-B2 PKC inhibitors for the treatment of septic cholestasis with polymethine dye targeting PRKCH, PRKCZ, PIKFYVE ACHE 4152/4885CHRM1 2671/4885ALDH1A1 4832/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.