SCHEMBL19554182

SCHEMBL19554182

O=C(Nc1cc(OC2COC2)c(F)cc1C(=O)O)c1ccc2cc(F)ccc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.42
ALB P02768 1/20 0.41
RAB9A P51151 3/20 0.40
BCL9 O00512 2/20 0.40
CTNNB1 P35222 2/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA7 P43166 1/20 0.39
KCNK2 O95069 1/20 0.39
DHODH Q02127 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PDE4D Q08499 1/20 0.38
AKR1C4 P17516 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19554215 0.90 SMN1; SMN2 (0.44) NPC1ALBRAB9ABCL9CTNNB1
SCHEMBL19554194 0.88 PDE5A (0.39) NPC1ALBBCL9CTNNB1CA12
SCHEMBL19554238 0.83 SERPINE1 (0.45) NPC1ALBRAB9ABCL9CTNNB1
SCHEMBL19554108 0.82 CYP1A2 (0.55) NPC1RAB9ACA12CA1CA7
SCHEMBL19554123 0.80 KCNK2 (0.50) NPC1RAB9AKCNK2DHODHCYP1A2
SCHEMBL19554233 0.79 HDAC3 (0.41) SMN1; SMN2
SCHEMBL19554214 0.79 BCL9 (0.38) BCL9CTNNB1CYP1A2CYP3A4CYP2C19
SCHEMBL19554158 0.78 SLC16A3 (0.46) NPC1RAB9ACA12CA1CA7
SCHEMBL19554122 0.77 AKR1C4 (0.61) NPC1RAB9ACA12CA1CA7
SCHEMBL19554254 0.77 HDAC3 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO claimed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed