SCHEMBL19554194

SCHEMBL19554194

N#Cc1cc(C(=O)O)c(NC(=O)c2ccc3cc(F)ccc3c2)cc1OC1COC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.39
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE1C Q14123 1/20 0.39
GPR6 P46095 4/20 0.38
BCL9 O00512 2/20 0.37
CTNNB1 P35222 2/20 0.37
SLC16A3 O15427 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA7 P43166 1/20 0.37
ALB P02768 1/20 0.36
KCNK2 O95069 1/20 0.36
DHODH Q02127 1/20 0.36
NPC1 O15118 1/20 0.35
GRM5 P41594 1/20 0.35
AKR1C4 P17516 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19554158 0.91 SLC16A3 (0.46) PDE5APDE1APDE1BPDE1CSLC16A3
SCHEMBL19554254 0.89 HDAC3 (0.40) GPR6GRM5
SCHEMBL19554182 0.88 NPC1 (0.42) BCL9CTNNB1CA12CA1CA7
SCHEMBL19554215 0.86 SMN1; SMN2 (0.44) BCL9CTNNB1CA12CA1CA7
SCHEMBL19554219 0.84 AKR1C4 (0.48) CA12CA1CA7NPC1AKR1C4
SCHEMBL19554178 0.81 NPC1 (0.52) NPC1AKR1C2AKR1C1
SCHEMBL19554262 0.80 KCNK2 (0.44) SLC16A3KCNK2DHODHNPC1AKR1C2
SCHEMBL19554171 0.79 PDE5A (0.48) PDE5APDE1APDE1BPDE1CAKR1C4
SCHEMBL19575809 0.78 KCNK2 (0.42) SLC16A3KCNK2DHODH
SCHEMBL19554185 0.78 RAB9A (0.44) SLC16A3KCNK2DHODHNPC1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO claimed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed