SCHEMBL19554249

SCHEMBL19554249

O=C(Nc1cc(-c2ccccc2F)c(Cl)cc1C(=O)O)c1ccc2cc(F)ccc2c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.50
PRSS12 P56730 2/20 0.46
DHODH Q02127 1/20 0.46
SERPINE1 P05121 5/20 0.44
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
PKM P14618 1/20 0.43
GRIK1 P39086 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HDAC1 Q13547 1/20 0.42
AKR1C4 P17516 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
AKR1C1 Q04828 1/20 0.41
ERO1A Q96HE7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19554330 0.85 KCNK2 (0.46) ACLYPRSS12DHODHMAPTMEN1
SCHEMBL19554126 0.84 PRSS12 (0.47) ACLYPRSS12DHODHSERPINE1MAPT
SCHEMBL19554240 0.83 STING1 (0.50) ACLYPRSS12DHODHMAPTMEN1
SCHEMBL19554248 0.82 ABL1 (0.48) ACLYPRSS12DHODHSERPINE1MAPT
SCHEMBL19554195 0.82 ABL1 (0.50) ACLYSERPINE1HDAC1
SCHEMBL19554172 0.81 DHODH (0.52) ACLYPRSS12DHODHSERPINE1MAPT
SCHEMBL19554123 0.80 KCNK2 (0.50) ACLYDHODHMAPTMEN1PKM
SCHEMBL19554229 0.79 SERPINE1 (0.61) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL19554338 0.79 SLC16A3 (0.43) ACLYDHODHSERPINE1MEN1PKM
SCHEMBL19554206 0.79 SLC16A3 (0.43) ACLYPRSS12DHODHMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO claimed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed