SCHEMBL19554352

SCHEMBL19554352

O=C(Nc1cc(F)c(F)cc1-c1nnn[nH]1)c1ccc2cc(F)ccc2c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 4/20 0.45
HDAC1 Q13547 1/20 0.40
HDAC3 O15379 3/20 0.39
HDAC2 Q92769 1/20 0.39
NPC1 O15118 6/20 0.39
RAB9A P51151 6/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GAA P10253 1/20 0.39
MAOB P27338 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CASP3 P42574 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
MLLT1 Q03111 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19554168 0.86 KCNMA1 (0.43) GPR35HDAC1HDAC3HDAC2NPC1
SCHEMBL19554687 0.78 KLKB1 (0.42) GPR35HDAC1HDAC3HDAC2NPC1
SCHEMBL1307013 0.75 KCNMA1 (0.56) GPR35HDAC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL19554341 0.74 HDAC3 (0.45) HDAC3NPC1RAB9ASMN1; SMN2
SCHEMBL1308878 0.73 GPR35 (0.55) GPR35NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL19554123 0.72 KCNK2 (0.50) HDAC1NPC1RAB9ASMN1; SMN2GAA
SCHEMBL4422766 0.72 GPR35 (0.52) GPR35HDAC1HDAC3HDAC2NPC1
SCHEMBL19554379 0.72 HDAC3 (0.40) GPR35HDAC1HDAC3HDAC2NPC1
SCHEMBL1307938 0.70 GPR35 (0.53) GPR35NPC1RAB9A
SCHEMBL1307860 0.69 GPR35 (0.56) GPR35HDAC1NPC1RAB9ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO claimed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed