SCHEMBL1961773

SCHEMBL1961773

COc1ccc(N)c(Oc2ccccc2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.63
CYP3A4 P08684 3/20 0.63
LTA4H P09960 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.53
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAPT P10636 2/20 0.48
THRB P10828 1/20 0.48
L3MBTL1 Q9Y468 3/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
CA4 P22748 1/20 0.46
GAA P10253 2/20 0.46
NPSR1 Q6W5P4 1/20 0.45
ADRA2B P18089 1/20 0.45
PTGS1 P23219 1/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18988645 0.90 ALDH1A1 (0.70) ALDH1A1CYP3A4LTA4HSMN1; SMN2MEN1
SCHEMBL5013387 0.86 MAOA (0.56) ALDH1A1CYP3A4LTA4HSMN1; SMN2MEN1
SCHEMBL9271567 0.85 ALDH1A1 (0.63) ALDH1A1CYP3A4LTA4HSMN1; SMN2MEN1
SCHEMBL5312459 0.85 ALDH1A1 (0.63) ALDH1A1CYP3A4LTA4HSMN1; SMN2MEN1
SCHEMBL1298542 0.85 ALDH1A1 (0.62) ALDH1A1CYP3A4LTA4HSMN1; SMN2MEN1
SCHEMBL18988688 0.84 ALDH1A1 (0.67) ALDH1A1CYP3A4SMN1; SMN2MEN1KMT2A
SCHEMBL1298894 0.83 ALDH1A1 (0.55) ALDH1A1CYP3A4LTA4HSMN1; SMN2MEN1
SCHEMBL11015595 0.81 CA12 (0.65) ALDH1A1CYP3A4LTA4HSMN1; SMN2MEN1
SCHEMBL11784875 0.81 CA12 (0.65) ALDH1A1CYP3A4LTA4HSMN1; SMN2MEN1
SCHEMBL76745 0.80 ALDH1A1 (0.95) ALDH1A1CYP3A4SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12384777-B2 Compounds comprising N-methyl-2-pyridone, and pharmaceutically acceptable salts Tay Therapeutics Limited (GB) 2025-08-12 US disclosed
CN-115356315-A Method for detecting hydrogen sulfide by fluorane derivative probe 沈阳感光化工研究院有限公司 2022-11-18 CN disclosed
US-20220204500-A1 COMPOUNDS COMPRISING N-METHYL-2-PYRIDONE, AND PHARMACEUTICALLY ACCEPTABLE SALTS UNIVERSITY OF DUNDEE (GB) 2022-06-30 US disclosed
US-20220204500-A1 COMPOUNDS COMPRISING N-METHYL-2-PYRIDONE, AND PHARMACEUTICALLY ACCEPTABLE SALTS UNIVERSITY OF DUNDEE (GB) 2022-06-30 US disclosed
CN-113924298-A Compounds comprising N-methyl-2-pyridone and pharmaceutically acceptable salts 邓迪大学 2022-01-11 CN disclosed
WO-2020216779-A1 COMPOUNDS COMPRISING N-METHYL-2-PYRIDONE, AND PHARMACEUTICALLY ACCEPTABLE SALTS UNIVERSITY OF DUNDEE (GB) 2020-10-29 WO disclosed
WO-2020216779-A1 COMPOUNDS COMPRISING N-METHYL-2-PYRIDONE, AND PHARMACEUTICALLY ACCEPTABLE SALTS UNIVERSITY OF DUNDEE (GB) 2020-10-29 WO disclosed
EP-1919892-B1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORP (US) 2013-08-14 EP disclosed
EP-1919892-B1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORP (US) 2013-08-14 EP disclosed
US-8481568-B2 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION (US) 2013-07-09 US disclosed
US-8481568-B2 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION (US) 2013-07-09 US disclosed
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SEPRACOR INC. 2011-06-16 US disclosed
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SEPRACOR INC. 2011-06-16 US disclosed
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SEPRACOR INC. 2011-06-16 US disclosed
EP-1919892-A2 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORPORATION (US) 2008-05-14 EP disclosed
WO-2007027527-A2 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORPORATION (US) 2007-03-08 WO disclosed
WO-2007027527-A2 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORPORATION (US) 2007-03-08 WO disclosed
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US disclosed
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US disclosed
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220204500-A1 COMPOUNDS COMPRISING N-METHYL-2-PYRIDONE, AND PHARMACEUTICALLY ACCEPTABLE SALTS TPMT, IL5, P2RY6 ALDH1A1 1800/4885CYP3A4 250/4885LTA4H 1389/4885
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SI, CYP3A5, CYP2D6 ALDH1A1 1081/4885CYP3A4 16/4885LTA4H 1719/4885
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same SI, CYP3A5, CYP2D6 ALDH1A1 1081/4885CYP3A4 16/4885LTA4H 1719/4885
US-12384777-B2 Compounds comprising N-methyl-2-pyridone, and pharmaceutically acceptable salts TPMT, IL5, P2RY6 ALDH1A1 1800/4885CYP3A4 250/4885LTA4H 1389/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.