SCHEMBL19617864

SCHEMBL19617864

C[Si](C)(C)CCOCC1CCc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.42
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
IDO1 P14902 2/20 0.38
PDPK1 O15530 1/20 0.38
BCHE P06276 2/20 0.36
MAOA P21397 3/20 0.36
MAOB P27338 3/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
ACHE P22303 1/20 0.36
ADRA1A P35348 1/20 0.36
SRD5A1 P18405 1/20 0.35
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10447649 0.80 HTR6 (0.47) HTR6MTNR1AMTNR1BIDO1PDPK1
SCHEMBL18025388 0.77 MTNR1A (0.48) HTR6MTNR1AMTNR1BPDPK1BCHE
SCHEMBL28768460 0.76 HTR6 (0.50) HTR6MTNR1AMTNR1BIDO1PDPK1
SCHEMBL22400816 0.74 CA2 (0.54) ADRA2BADRA2C
SCHEMBL7680750 0.73 HTR6 (0.42) HTR6MTNR1AMTNR1BIDO1PDPK1
SCHEMBL7677975 0.73 HTR6 (0.44) HTR6MTNR1AMTNR1BIDO1PDPK1
SCHEMBL10447102 0.71 IDO1 (0.46) IDO1
SCHEMBL9115029 0.70 HTR6 (0.54) HTR6MTNR1AMTNR1BIDO1PDPK1
SCHEMBL14143008 0.70 CA2 (0.45) HTR6MTNR1AMTNR1BIDO1PDPK1
SCHEMBL6978852 0.70 CA2 (0.45) HTR6MTNR1AMTNR1BIDO1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458445-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2019-03-27 EP disclosed
WO-2017201161-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2017-11-23 WO disclosed