SCHEMBL19632148

SCHEMBL19632148

CC(C)OCCN1CCN(C2(C(O)c3ccccn3)CC(C)(C)OC(C)(C)C2)CC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
SLC6A2 P23975 1/20 0.35
DRD2 P14416 1/20 0.35
KDM1A O60341 1/20 0.35
LTA4H P09960 1/20 0.34
PTGS2 P35354 1/20 0.34
GAA P10253 1/20 0.34
OPRM1 P35372 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
ALDH1A1 P00352 1/20 0.33
IDH1 O75874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19632043 0.79 DRD2 (0.36) DRD2LTA4HPTGS2GAAOPRM1
SCHEMBL19631944 0.78 GRM4 (0.37) SLC6A4SLC6A3SLC6A2DRD2OPRM1
SCHEMBL22169640 0.78 OPRM1 (0.37) DRD2LTA4HPTGS2GAAOPRM1
SCHEMBL21233604 0.71 CHRM2 (0.41) DRD2OPRM1ALDH1A1IDH1
SCHEMBL19631833 0.71 SIGMAR1 (0.41) OPRM1SIGMAR1ALDH1A1
SCHEMBL19631794 0.70 OPRM1 (0.39) DRD2OPRM1SIGMAR1
SCHEMBL19631776 0.70 OPRM1 (0.39) DRD2OPRM1SIGMAR1
SCHEMBL19631779 0.70 OPRM1 (0.39) DRD2OPRM1SIGMAR1
SCHEMBL18425135 0.70 OPRM1 (0.39) SLC6A4SLC6A3SLC6A2DRD2OPRM1
SCHEMBL20482028 0.70 ALDH1A1 (0.39) DRD2SIGMAR1ALDH1A1IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed