SCHEMBL19632043

SCHEMBL19632043

COCCN1CCN(C2(C(O)c3ccccn3)CCOC(C)(C)C2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.36
ACHE P22303 2/20 0.34
KCNA5 P22460 1/20 0.34
OPRM1 P35372 2/20 0.34
DRD3 P35462 1/20 0.34
LTA4H P09960 1/20 0.33
PTGS2 P35354 1/20 0.33
GAA P10253 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
IDH1 O75874 1/20 0.33
HTT P42858 1/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22169640 0.89 OPRM1 (0.37) DRD2OPRM1DRD3LTA4HPTGS2
SCHEMBL19631833 0.85 SIGMAR1 (0.41) OPRM1ALDH1A1KDM4ESIGMAR1SMN1; SMN2
SCHEMBL22169613 0.83 DRD2 (0.35) DRD2OPRM1DRD3ALDH1A1KDM4E
SCHEMBL22169548 0.81 SIGMAR1 (0.40) OPRM1ALDH1A1SIGMAR1TSHRSMN1; SMN2
SCHEMBL19632148 0.79 SLC6A4 (0.35) DRD2OPRM1LTA4HPTGS2GAA
SCHEMBL19632060 0.77 HTR1A (0.40) DRD2OPRM1DRD3GAAKDM4E
SCHEMBL21233604 0.74 CHRM2 (0.41) DRD2KCNA5OPRM1DRD3ALDH1A1
SCHEMBL19631835 0.71 LMNA (0.35) OPRM1ALDH1A1KDM4ESIGMAR1HTT
SCHEMBL20482028 0.70 ALDH1A1 (0.39) DRD2KCNA5DRD3ALDH1A1SIGMAR1
SCHEMBL19631794 0.69 OPRM1 (0.39) DRD2OPRM1DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed