SCHEMBL19633643

SCHEMBL19633643

COc1cc([N+](=O)[O-])ccc1Nc1ccnc2cc(OCCCc3ccccc3)ccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.49
KMT2A Q03164 6/20 0.49
MEN1 O00255 5/20 0.49
CYP19A1 P11511 4/20 0.49
CYP11B1 P15538 3/20 0.49
CYP11B2 P19099 3/20 0.49
CCNC P24863 1/20 0.48
CDK8 P49336 1/20 0.48
LMNA P02545 2/20 0.46
ALDH1A1 P00352 2/20 0.45
HTT P42858 1/20 0.45
KDM4E B2RXH2 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
PKM P14618 1/20 0.43
POLB P06746 1/20 0.43
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633815 0.93 MEN1 (0.51) MAPTKMT2AMEN1CYP19A1CYP11B1
SCHEMBL19633692 0.85 CCNC (0.50) MAPTKMT2AMEN1CYP19A1CYP11B1
SCHEMBL19633545 0.84 KMT2A (0.49) KMT2AMEN1CYP19A1CYP11B1CYP11B2
SCHEMBL19633797 0.76 CYP19A1 (0.47) MAPTKMT2AMEN1CYP19A1CYP11B1
SCHEMBL19633503 0.76 GAK (0.53) HTTGAKRIPK2COQ8ANLK
SCHEMBL19633549 0.74 KMT2A (0.55) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL1157681 0.73 CYP19A1 (0.62) MAPTKMT2AMEN1CYP19A1CYP11B1
SCHEMBL19633574 0.73 CTSV (0.56) MAPTKMT2AMEN1CCNCCDK8
SCHEMBL26086283 0.73 GAK (0.59) ALDH1A1POLBGAKRIPK2COQ8A
SCHEMBL19633777 0.73 GAK (0.57) KMT2ALMNAALDH1A1GAKRIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed