SCHEMBL19633683

SCHEMBL19633683

COc1cccc(Sc2ccnc3cc(OCCCc4ccccc4)ccc23)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
TLR8 Q9NR97 1/20 0.41
HTR1A P08908 2/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
EGFR P00533 1/20 0.40
CYP1A2 P05177 1/20 0.40
SLC2A1 P11166 1/20 0.40
MET P08581 1/20 0.40
PDGFRA P16234 1/20 0.40
KDR P35968 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
MAOB P27338 2/20 0.39
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633750 0.87 MAOA (0.39) METKDRCYP11B1CYP11B2MAOB
SCHEMBL19633646 0.87 MAOB (0.39) MAOBMAOAGRM4
SCHEMBL19633857 0.87 CYP4F2 (0.42) CYP3A4ADRA1DADRA1AADRA1BKDR
SCHEMBL19633520 0.83 MAOB (0.46) CYP3A4TLR8HTR1AADRA1DADRA1A
SCHEMBL200813 0.82 PDGFRA (0.53) CYP3A4TLR8HTR1AADRA1DADRA1A
SCHEMBL19633645 0.79 SLC6A2 (0.43) MAOBMAOAGRM4
SCHEMBL19633753 0.79 GAK (0.49) CYP3A4TLR8HTR1AADRA1DADRA1A
SCHEMBL19633648 0.79 PDGFRA (0.46) TLR8HTR1AADRA1DADRA1AADRA1B
SCHEMBL19633503 0.78 GAK (0.53) HTR1AADRA1DADRA1AADRA1BEGFR
SCHEMBL7487186 0.77 KDR (0.58) EGFRPDGFRAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed