SCHEMBL19634802

SCHEMBL19634802

CC(=O)NCc1cccc(C(=O)NCCN(C)C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.53
MRGPRX4 Q96LA9 1/20 0.51
ROCK2 O75116 2/20 0.50
MMP13 P45452 1/20 0.49
PKM P14618 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPK1 P28482 1/20 0.48
ROCK1 Q13464 1/20 0.47
LMNA P02545 2/20 0.47
TP53 P04637 2/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22754705 0.88 PARP1 (0.54) PARP1MRGPRX4ROCK2MMP13PKM
SCHEMBL23471351 0.87 ALDH1A1 (0.55) ROCK2MMP13ALDH1A1MAPK1LMNA
SCHEMBL21015872 0.86 MRGPRX4 (0.51) PARP1MRGPRX4ROCK2MMP13PKM
SCHEMBL12333454 0.85 USP2 (0.55) PARP1MRGPRX4PKMALDH1A1MAPK1
SCHEMBL16380331 0.85 ROCK2 (0.53) ROCK2MMP13ALDH1A1ROCK1LMNA
SCHEMBL5109753 0.83 LOXL2 (0.54) PARP1MRGPRX4PKMALDH1A1MAPK1
SCHEMBL23470991 0.83 HDAC1 (0.62) ALDH1A1HDAC3HDAC4HDAC1HDAC2
SCHEMBL23889139 0.82 SMN1; SMN2 (0.54) PARP1MRGPRX4ROCK2PKMALDH1A1
SCHEMBL19634816 0.82 ROCK2 (0.57) MRGPRX4ROCK2MMP13ROCK1LMNA
SCHEMBL19634746 0.81 MMP13 (0.49) ROCK2MMP13ALDH1A1ROCK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed