SCHEMBL19635384

SCHEMBL19635384

OCCn1nc(C2CC2)c(Br)c1CO

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.42
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
CSNK2A1 P68400 1/20 0.33
CSNK2A3 Q8NEV1 1/20 0.33
PDE10A Q9Y233 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19635547 0.83 EPHX2 (0.33) EPHX2PDE10A
SCHEMBL19615303 0.83 ALDH1A1 (0.34) EPHX2PDE10A
SCHEMBL6166773 0.65 HTT (0.52) EPHX2
SCHEMBL17594894 0.63 MPO (0.43) PDE10A
SCHEMBL21889237 0.59 AOC3 (0.39) PDE10A
SCHEMBL11629541 0.58 CSNK2A2 (0.41) CSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL17045428 0.58 NPC1 (0.40) EPHX2PDE10A
SCHEMBL19635867 0.57
SCHEMBL21301526 0.56 PDE10A (0.52) EPHX2PDE10A
SCHEMBL6920216 0.56 APAF1 (0.50) CSNK2A2CSNK2BCSNK2A1CSNK2A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed