SCHEMBL19664706

SCHEMBL19664706

O=C(O)CC(c1ccccc1)c1ccncn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 1/20 0.41
GABBR1 Q9UBS5 1/20 0.41
CTSA P10619 2/20 0.41
FFAR1 O14842 1/20 0.40
EPHX2 P34913 1/20 0.40
CASP1 P29466 1/20 0.40
LMNA P02545 3/20 0.39
HMOX2 P30519 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
TBXAS1 P24557 1/20 0.38
ALPL P05186 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28788265 0.83 ALDH1A1 (0.43) CASP1LMNACYP2C19ALDH1A1CYP3A4
SCHEMBL1131686 0.81 ALDH1A1 (0.55) GABBR2GABBR1FFAR1EPHX2CASP1
SCHEMBL170301 0.79 SLC6A2 (0.55) GABBR2GABBR1FFAR1EPHX2LMNA
SCHEMBL1888807 0.78 GABBR2 (0.44) GABBR2GABBR1CTSAFFAR1LMNA
SCHEMBL22408433 0.78 AHR (0.37) CTSAFFAR1ALDH1A1TSHRKDM4E
Hydrochloric Acid SCHEMBL128794 0.78 SLC6A2 (0.53) GABBR2GABBR1FFAR1EPHX2LMNA
SCHEMBL16150460 0.77 P2RX7 (0.42) GABBR2GABBR1PTGDR2CYP2C19CYP3A4
SCHEMBL28092231 0.77 L3MBTL1 (0.41) PTGDR2CYP2C19ALDH1A1TSHRKDM4E
SCHEMBL21643045 0.76 CTSA (0.52) CTSA
SCHEMBL4557709 0.74 ALDH1A1 (0.44) LMNASLC6A2SLC6A4SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091940-B3 4-PHENYL-6-(2,2,2-TRIFLUORO-1-PHENYLETHOXY)PYRIMIDINE-BASED COMPOUNDS AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS INC (US) 2017-12-06 EP disclosed