SCHEMBL19669654

SCHEMBL19669654

C=C(C)CN1C(=O)COc2cc(NC(C)=O)ccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.51
ALOX15 P16050 3/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 3/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
RORC P51449 1/20 0.46
PLK1 P53350 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
OPRK1 P41145 1/20 0.45
UTS2R Q9UKP6 1/20 0.45
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19669631 0.86 RORC (0.57) TSHRALOX15POLBMAPTKDM4E
SCHEMBL17996431 0.86 TP53 (0.53) TSHRALOX15POLBMAPTKDM4E
SCHEMBL18010766 0.85 TSHR (0.43) TSHRALOX15POLBMAPTKDM4E
SCHEMBL19669648 0.85 TSHR (0.45) TSHRALOX15POLBMAPTKDM4E
SCHEMBL19669647 0.81 ITGB3 (0.63) ITGB3ITGA2B
SCHEMBL19669650 0.81 NOS3 (0.51) TSHRALOX15POLBMAPTKDM4E
SCHEMBL19669652 0.80 CYP1A2 (0.52) TSHRPOLBMAPTALDH1A1CYP1A2
SCHEMBL17996374 0.80 MAPT (0.59) TSHRALOX15POLBMAPTALDH1A1
SCHEMBL19669633 0.80 CYP3A4 (0.52) TSHRPOLBMAPTKDM4ECYP1A2
SCHEMBL19669656 0.80 ITGB3 (0.54) MAPTKDM4EALDH1A1GAARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9834520-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-12-05 US disclosed