SCHEMBL19669739

SCHEMBL19669739

CC(C)(C)NC(=O)/C=C/CN1CCN(S(C)(=O)=O)CC1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 2/20 0.35
PKM P14618 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
ATM Q13315 1/20 0.34
POLB P06746 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
MAPT P10636 1/20 0.33
TP53 P04637 1/20 0.33
LMNA P02545 2/20 0.32
EGFR P00533 1/20 0.32
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15600777 0.85 TDP1 (0.38) ALDH1A1KDM4ETDP1ATMNPSR1
SCHEMBL19912771 0.82 PKM (0.36) ALDH1A1KDM4EPKMLMNAEGFR
SCHEMBL19669740 0.82 LMNA (0.38) ALDH1A1KDM4ELMNAEGFR
SCHEMBL19912779 0.82 SMN1; SMN2 (0.45) ALDH1A1LMNAEGFR
SCHEMBL24637162 0.81 EGFR (0.34) ALDH1A1LMNAEGFR
SCHEMBL19442308 0.80 SMN1; SMN2 (0.47) ALDH1A1LMNAEGFR
SCHEMBL19669738 0.79 SMN1; SMN2 (0.38) ALDH1A1KDM4EPOLBTP53LMNA
SCHEMBL15600836 0.78 SIGMAR1 (0.41) ALDH1A1KDM4EPKMLMNAEGFR
SCHEMBL15600841 0.78 SMN1; SMN2 (0.53) ALDH1A1KDM4EEGFRTSHR
SCHEMBL20235763 0.77 ACKR3 (0.35) ALDH1A1LMNAEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9834571-B2 Compounds for inhibiting cell proliferation in EGFR-driven cancers ARIAD PHARMACEUTICALS, INC. (US) 2017-12-05 US disclosed