SCHEMBL19676366

SCHEMBL19676366

CONc1ccc(Oc2cccnc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.53
TDP1 Q9NUW8 2/20 0.53
CYP19A1 P11511 2/20 0.53
ALDH1A1 P00352 3/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
HTT P42858 2/20 0.52
GAA P10253 1/20 0.52
HPGD P15428 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.49
TTBK1 Q5TCY1 1/20 0.48
TTBK2 Q6IQ55 1/20 0.48
TP53 P04637 1/20 0.48
RECQL P46063 1/20 0.48
LTA4H P09960 1/20 0.48
KDM4E B2RXH2 2/20 0.47
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
MAPT P10636 1/20 0.46
NAMPT P43490 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13232649 0.83 LMNA (0.56) LMNATDP1CYP19A1ALDH1A1NPC1
SCHEMBL16114401 0.82 LMNA (0.75) LMNATDP1CYP19A1ALDH1A1NPC1
SCHEMBL11107948 0.80 LMNA (0.62) LMNATDP1CYP19A1ALDH1A1NPC1
SCHEMBL20041022 0.80 HPGD (0.61) ALDH1A1NPC1RAB9AHTTHPGD
SCHEMBL13707699 0.79 LMNA (0.56) LMNATDP1CYP19A1ALDH1A1NPC1
SCHEMBL25000186 0.79 LMNA (0.51) LMNATDP1CYP19A1ALDH1A1NPC1
SCHEMBL22874526 0.79 TDP1 (0.51) LMNATDP1CYP19A1ALDH1A1NPC1
Hydrochloric Acid SCHEMBL4374994 0.78 LMNA (0.55) LMNATDP1CYP19A1ALDH1A1NPC1
SCHEMBL27968872 0.78 LMNA (0.69) LMNATDP1CYP19A1ALDH1A1NPC1
SCHEMBL676142 0.78 LMNA (0.82) LMNATDP1CYP19A1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080098-B1 INHIBITORS OF BRUTON'S TYROSINE KINASE HOFFMANN LA ROCHE (CH) 2017-12-06 EP disclosed