SCHEMBL19684412

SCHEMBL19684412

CCN/C(=C(\C(=O)Nc1cccc(C(F)(F)F)c1)C(=O)OCC)c1ccnn1-c1ccc(C#N)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ELANE P08246 9/20 0.43
IDH1 O75874 1/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
AURKA O14965 1/20 0.39
BRAF P15056 1/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
ALOX12 P18054 1/20 0.39
ATM Q13315 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.38
SAE1 Q9UBE0 1/20 0.38
UBA2 Q9UBT2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19684403 0.93 ELANE (0.47) ELANEIDH1CYP3A4CYP2C9AURKA
SCHEMBL19684522 0.83 ELANE (0.48) ELANEIDH1AURKAMAPTRXFP1
SCHEMBL19684419 0.82 ELANE (0.48) ELANEIDH1AURKAMAPTRXFP1
SCHEMBL19688572 0.81 BRAF (0.37) ELANEIDH1BRAFGAAMAPT
SCHEMBL19684417 0.76 UBE2M (0.42) ELANEAURKASMN1; SMN2MEN1KMT2A
SCHEMBL19684414 0.76 ELANE (0.41) ELANEIDH1AURKARXFP1MEN1
SCHEMBL19640137 0.75 ELANE (0.46) ELANEIDH1CYP3A4CYP2C9AURKA
SCHEMBL19640095 0.74 ELANE (0.49) ELANEIDH1AURKAMAPTRXFP1
SCHEMBL19640079 0.73 ELANE (0.47) ELANEIDH1CYP2C9AURKAGAA
SCHEMBL19640140 0.71 ELANE (0.43) ELANECYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017207432-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2017-12-07 WO disclosed