SCHEMBL19684419

SCHEMBL19684419

CN/C(=C(/C(C)=O)C(=O)Nc1cccc(C(F)(F)F)c1)c1ccnn1-c1ccc(C#N)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.48
AURKA O14965 1/20 0.42
RXFP1 Q9HBX9 2/20 0.42
IDH1 O75874 1/20 0.42
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
SAE1 Q9UBE0 1/20 0.39
UBA2 Q9UBT2 1/20 0.39
NPC1 O15118 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 1/20 0.38
KCNJ6 P48051 1/20 0.38
KCNJ5 P48544 1/20 0.38
KCNJ3 P48549 1/20 0.38
KLKB1 P03952 1/20 0.37
KIT P10721 1/20 0.37
DDR1 Q08345 1/20 0.37
DDR2 Q16832 1/20 0.37
LDHA P00338 1/20 0.37
NPY5R Q15761 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19684522 0.94 ELANE (0.48) ELANEAURKARXFP1IDH1KDM4E
SCHEMBL19684403 0.90 ELANE (0.47) ELANEAURKARXFP1IDH1KDM4E
SCHEMBL19684417 0.86 UBE2M (0.42) ELANEAURKANPC1SMN1; SMN2KLKB1
SCHEMBL19684414 0.84 ELANE (0.41) ELANEAURKARXFP1IDH1KCNJ6
SCHEMBL19684412 0.82 ELANE (0.43) ELANEAURKARXFP1IDH1KDM4E
SCHEMBL19640095 0.77 ELANE (0.49) ELANEAURKARXFP1IDH1KDM4E
SCHEMBL19684716 0.77 MAPT (0.43) ELANEAURKARXFP1IDH1KDM4E
SCHEMBL19640079 0.77 ELANE (0.47) ELANEAURKARXFP1IDH1KDM4E
SCHEMBL19688572 0.76 BRAF (0.37) ELANEIDH1KDM4EMAPTSMN1; SMN2
SCHEMBL19640137 0.75 ELANE (0.46) ELANEAURKARXFP1IDH1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017207432-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2017-12-07 WO disclosed