SCHEMBL19700360

SCHEMBL19700360

CC(C)(C)S(=O)(=O)NC1CCC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.46
CA7 P43166 3/20 0.46
CA14 Q9ULX7 3/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.39
KDM4E B2RXH2 1/20 0.39
RECQL P46063 1/20 0.39
NPY5R Q15761 1/20 0.38
ALDH1A1 P00352 5/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
HPGD P15428 1/20 0.36
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16230729 0.95 CA12 (0.52) CA12CA7CA14CA1CA2
SCHEMBL13958956 0.93 CA1 (0.56) CA12CA7CA14CA1CA2
SCHEMBL12855687 0.93 CA1 (0.56) CA12CA7CA14CA1CA2
SCHEMBL12048931 0.90 CA12 (0.50) CA12CA7CA14CA1CA2
SCHEMBL14314445 0.82 CA12 (0.42) CA12CA7CA14CA1CA2
SCHEMBL13054260 0.82 CA12 (0.42) CA12CA7CA14CA1CA2
SCHEMBL10133146 0.82 CA12 (0.42) CA12CA7CA14CA1CA2
SCHEMBL13204637 0.80 EPHX1 (0.39) CA12CA7CA14CA1NPY5R
SCHEMBL13113463 0.79 NPY5R (0.37) CA12CA7CA14CA1NPY5R
SCHEMBL23758147 0.78 BRD4 (0.41) CA12CA7CA14CA1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230250095-A1 BENZIMIDAZOLE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF TUOJIE BIOTECH(SHANGHAI) CO., LTD. (CN) 2023-08-10 US disclosed
US-20230250095-A1 BENZIMIDAZOLE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF TUOJIE BIOTECH(SHANGHAI) CO., LTD. (CN) 2023-08-10 US disclosed
US-11236111-B2 Hepatitis B antiviral agents ENANTA PHARMACEUTICALS, INC. (US) 2022-02-01 US disclosed
US-10975088-B2 Imidazo[2,1-f][1,2,4]triazine compounds as pi3k-y inhibitors INCYTE CORPORATION (US) 2021-04-13 US disclosed
US-20210047312-A1 INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE GAMMA ASTRAZENECA AB (SE) 2021-02-18 US disclosed
US-20200385391-A1 HEPATITIS B ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2020-12-10 US disclosed
US-10858355-B2 Inhibitors of phosphatidylinositol 3-kinase gamma ASTRAZENECA AB (SE) 2020-12-08 US disclosed
US-20200377519-A1 HEPATITIS B ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2020-12-03 US disclosed
US-20200317678-A1 HEPATITIS B ANTIVIRAL AGENTS ENANTA PHARM INC (US) 2020-10-08 US disclosed
US-20200299289-A1 NOVEL INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE GAMMA ASTRAZENECA AB (SE) 2020-09-24 US disclosed
US-10640511-B2 Hepatitis B antiviral agents Enant Pharmaceuticals, Inc. (US) 2020-05-05 US disclosed
US-10428070-B2 Hepatitis B antiviral agents ENANTA PHARMACEUTICALS, INC. (US) 2019-10-01 US disclosed
US-20190177320-A1 HEPATITIS B ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2019-06-13 US disclosed
US-20190119288-A1 HEPATITIS B ANTIVIRAL AGENTS ENANTA PHARM INC (US) 2019-04-25 US disclosed
US-10189846-B2 Hepatitis B antiviral agents ENANTA PHARMACEUTICALS, INC. (US) 2019-01-29 US disclosed
US-20180009816-A1 HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS INCYTE CORPORATION 2018-01-11 US disclosed
US-20170355701-A1 HEPATITIS B ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2017-12-14 US disclosed
US-20170355701-A1 HEPATITIS B ANTIVIRAL AGENTS ENANTA PHARMACEUTICALS, INC. 2017-12-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (16 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210047312-A1 INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE GAMMA PIK3CD, PIK3CG, PIK3CA CA12 4724/4885CA7 4040/4885CA14 4707/4885
US-11236111-B2 Hepatitis B antiviral agents HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-20190119288-A1 HEPATITIS B ANTIVIRAL AGENTS HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-20230250095-A1 BENZIMIDAZOLE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF P2RX7, P2RX3, P2RX5 CA12 4849/4885CA7 3498/4885CA14 4688/4885
US-20200385391-A1 HEPATITIS B ANTIVIRAL AGENTS HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-20200317678-A1 HEPATITIS B ANTIVIRAL AGENTS HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-20190177320-A1 HEPATITIS B ANTIVIRAL AGENTS HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-10189846-B2 Hepatitis B antiviral agents HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-10428070-B2 Hepatitis B antiviral agents HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-10858355-B2 Inhibitors of phosphatidylinositol 3-kinase gamma PIK3CD, PIK3CG, PIK3CA CA12 4724/4885CA7 4040/4885CA14 4707/4885
US-20200377519-A1 HEPATITIS B ANTIVIRAL AGENTS HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-20200299289-A1 NOVEL INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE GAMMA PI4KA, PIK3CD, PI4KB CA12 4747/4885CA7 3777/4885CA14 4652/4885
US-20170355701-A1 HEPATITIS B ANTIVIRAL AGENTS HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885
US-10975088-B2 Imidazo[2,1-f][1,2,4]triazine compounds as pi3k-y inhibitors PIK3R5, PIK3CD, PIK3CA CA12 4422/4885CA7 3039/4885CA14 4520/4885
US-20180009816-A1 HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS PIK3R5, PIK3CA, PIK3CD CA12 4623/4885CA7 2700/4885CA14 4554/4885
US-10640511-B2 Hepatitis B antiviral agents HAVCR2, SLC10A1, HDGF CA12 2997/4885CA7 3147/4885CA14 3206/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.