SCHEMBL19783854

SCHEMBL19783854

O=c1cnn(-c2ccc3nn(-c4cccnc4)cc3c2)c(=O)n1S

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.38
ESR2 Q92731 1/20 0.36
CYP2A6 P11509 1/20 0.34
CYP11B2 P19099 1/20 0.34
GRM1 Q13255 1/20 0.32
EP300 Q09472 1/20 0.32
KAT2B Q92831 1/20 0.32
USP8 P40818 1/20 0.32
MTOR P42345 2/20 0.31
PDE10A Q9Y233 1/20 0.31
HTT P42858 2/20 0.31
ALOX12 P18054 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21422259 0.87 ESR2 (0.39) TLR8ESR2CYP2A6CYP11B2GRM1
SCHEMBL19783858 0.87 TLR8 (0.45) TLR8ESR2CYP2A6CYP11B2GRM1
SCHEMBL19784106 0.86 TLR8 (0.38) TLR8ESR2CYP2A6CYP11B2GRM1
SCHEMBL19783977 0.86 ESR2 (0.41) TLR8ESR2CYP2A6CYP11B2GRM1
SCHEMBL19783976 0.84 ADORA2A (0.39) TLR8ESR2CYP2A6CYP11B2GRM1
SCHEMBL19783274 0.84 TLR8 (0.38) TLR8CYP2A6CYP11B2GRM1EP300
SCHEMBL19783853 0.84 CYP11B2 (0.37) ESR2CYP11B2
SCHEMBL19784142 0.83 TLR8 (0.35) TLR8CYP2A6CYP11B2GRM1EP300
SCHEMBL19783867 0.82 CYP11B2 (0.37) TLR8ESR2CYP2A6CYP11B2GRM1
SCHEMBL19783974 0.82 POLB (0.38) TLR8ESR2CYP2A6CYP11B2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3484877-B1 BICYCLIC COMPOUNDS AS PEST CONTROLLERS BAYER CROPSCIENCE AG (DE) 2020-07-01 EP disclosed
WO-2018011111-A1 BICYCLIC COMPOUNDS AS PEST CONTROL AGENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-01-18 WO disclosed