SCHEMBL19785591

SCHEMBL19785591

Cc1c(N)cc(Cl)cc1CN1CCN(C(=O)OC(C)C)CC1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MGLL Q99685 15/20 0.42
ABHD6 Q9BV23 6/20 0.42
PLA2G7 Q13093 5/20 0.42
KDM4E B2RXH2 2/20 0.41
TSHR P16473 1/20 0.41
POLB P06746 1/20 0.39
MTNR1B P49286 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19785782 0.88 MGLL (0.41) ALDH1A1MGLLABHD6PLA2G7KDM4E
SCHEMBL19785787 0.84 MGLL (0.41) ALDH1A1MGLLABHD6PLA2G7KDM4E
SCHEMBL19785873 0.84 VEGFA (0.51) ALDH1A1MGLLABHD6PLA2G7KDM4E
SCHEMBL29613591 0.83 PTGDR2 (0.44)
SCHEMBL19785590 0.83 PTGDR2 (0.44)
SCHEMBL19785970 0.82 CTSB (0.45) ALDH1A1MGLLABHD6PLA2G7KDM4E
SCHEMBL22383724 0.77 GRIN2B (0.55) ALDH1A1KDM4ETSHR
SCHEMBL18658594 0.77 RORC (0.55) ALDH1A1KDM4ETSHRMTNR1B
SCHEMBL20614093 0.76 ALDH1A1 (0.48) ALDH1A1KDM4EPOLB
SCHEMBL30642978 0.74 RORC (0.49) ALDH1A1KDM4ETSHRMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3484880-B1 HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA AS (DK) 2020-09-02 EP disclosed
WO-2018011201-A1 HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2018-01-18 WO disclosed