SCHEMBL19785970

SCHEMBL19785970

Cc1c(CN2CCN(C(=O)OC(C)C)CC2)cc(Cl)cc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.45
ALDH1A1 P00352 8/20 0.42
KDM4E B2RXH2 6/20 0.42
TDP1 Q9NUW8 2/20 0.42
LMNA P02545 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MGLL Q99685 5/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
BLM P54132 1/20 0.40
ABHD6 Q9BV23 3/20 0.40
PLA2G7 Q13093 2/20 0.40
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19785987 0.85 CTSB (0.46) CTSBALDH1A1KDM4ETDP1LMNA
SCHEMBL18658598 0.85 VEGFA (0.48) CTSBALDH1A1KDM4ETDP1LMNA
SCHEMBL21368976 0.84 PTGDR2 (0.42) ALDH1A1LMNAMEN1KMT2A
SCHEMBL29613545 0.84 PTGDR2 (0.42) ALDH1A1LMNAMEN1KMT2A
SCHEMBL19785591 0.82 ALDH1A1 (0.44) ALDH1A1KDM4EMGLLABHD6PLA2G7
SCHEMBL30643025 0.76 MEN1 (0.50) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL29133046 0.76 MEN1 (0.50) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL19785782 0.73 MGLL (0.41) ALDH1A1KDM4EMGLLABHD6PLA2G7
SCHEMBL21354265 0.72 PTGDR2 (0.46) ALDH1A1KDM4ETDP1MEN1KMT2A
SCHEMBL19785985 0.72 ALDH1A1 (0.45) CTSBALDH1A1KDM4ETDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3484880-B1 HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA AS (DK) 2020-09-02 EP disclosed
WO-2018011201-A1 HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2018-01-18 WO disclosed