SCHEMBL19791547

SCHEMBL19791547

Cc1ccc(F)c(-c2cc(-c3cncc(-c4noc(C5CCN(C)CC5)n4)c3)c3cccnc3n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.38
TSHR P16473 4/20 0.38
PPARA Q07869 1/20 0.38
CNR2 P34972 3/20 0.38
CASP3 P42574 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
HTT P42858 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
ALDH1A1 P00352 2/20 0.37
TP53 P04637 1/20 0.37
ALOX15 P16050 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440268 0.93 CNR2 (0.41) LMNATSHRPPARACNR2HTT
SCHEMBL2326924 0.91 CNR2 (0.45) LMNATSHRPPARACNR2HTT
SCHEMBL12440209 0.81 MET (0.43)
SCHEMBL12439728 0.78 MAPT (0.37) LMNATSHRALDH1A1ALOX15MAPK1
SCHEMBL12440225 0.78 GPR119 (0.44) CNR2HTTSMN1; SMN2TUBB4ATUBB
SCHEMBL2324592 0.77 LMNA (0.36) LMNATSHRHTTSMN1; SMN2ALDH1A1
SCHEMBL19791515 0.76 TLR9 (0.35)
SCHEMBL12439733 0.74 MET (0.46)
SCHEMBL12441209 0.74 MET (0.47)
SCHEMBL13968443 0.73 IDO1 (0.35) LMNATSHRHTTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531500-B1 HETARYL-[1,8]NAPHTHYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 2018-01-24 EP disclosed