SCHEMBL1980365

SCHEMBL1980365

COc1ccc2[nH]c3cnc(-c4cccnc4)cc3c2c1-c1ccc(C(=O)NCCC2CCCN2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 4/20 0.52
TLR9 Q9NR96 3/20 0.52
TLR8 Q9NR97 3/20 0.52
BRAF P15056 1/20 0.45
EGLN1 Q9GZT9 2/20 0.44
PTAFR P25105 2/20 0.39
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNB3 Q05901 1/20 0.38
WNT1 P04628 3/20 0.38
DYRK1A Q13627 3/20 0.38
ACKR3 P25106 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
PDE4B Q07343 1/20 0.37
NMT1 P30419 1/20 0.37
CHEK1 O14757 1/20 0.37
ACHE P22303 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979171 0.90 WNT1 (0.42) TLR7TLR9TLR8PTAFRWNT1
SCHEMBL1979088 0.87 WNT1 (0.51) TLR7TLR9TLR8WNT1DYRK1A
SCHEMBL1980360 0.87 KMT2A (0.48)
SCHEMBL1979499 0.87 KMT2A (0.48)
SCHEMBL12598121 0.86 KDM4E (0.44) TLR7TLR9TLR8WNT1DYRK1A
SCHEMBL12598125 0.86 DRD2 (0.48) TLR7TLR9TLR8PTAFRWNT1
SCHEMBL1983761 0.85 BRAF (0.47) TLR7TLR9BRAFPTAFRWNT1
SCHEMBL473719 0.85 BRAF (0.47) TLR7TLR9TLR8BRAFEGLN1
SCHEMBL1981803 0.85 MTNR1A (0.45) TLR7TLR9TLR8BRAFPTAFR
SCHEMBL12597820 0.84 TLR9 (0.40) TLR7TLR9TLR8CHRNB1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed