SCHEMBL19853693

SCHEMBL19853693

NC(=O)CN1CC2(CCN(OCc3ccccc3)CC2)C1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.48
ALDH1A1 P00352 2/20 0.38
OPRM1 P35372 4/20 0.38
OPRL1 P41146 4/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KMT2A Q03164 1/20 0.36
CYP2D6 P10635 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC8 Q9BY41 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
CXCR3 P49682 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
TSHR P16473 1/20 0.34
CRBN Q96SW2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19853733 0.83 DPP4 (0.47) RIPK1OPRM1OPRL1CYP2C19SMN1; SMN2
SCHEMBL19853697 0.77 RIPK1 (0.37) RIPK1ALDH1A1CYP2C19SMN1; SMN2KMT2A
SCHEMBL19853782 0.76 RIPK1 (0.51) RIPK1OPRM1OPRL1KMT2ACHRM2
SCHEMBL19853771 0.76 GRIN2B (0.41) RIPK1ALDH1A1OPRM1CYP2C19SMN1; SMN2
SCHEMBL17359168 0.70 CYP2C19 (0.42) CYP2C19SMN1; SMN2KMT2A
SCHEMBL9290068 0.70 DHFR (0.43) ALDH1A1OPRL1CYP2C19SMN1; SMN2NPC1
SCHEMBL19853789 0.70 APEX1 (0.47) RIPK1OPRM1OPRL1RAB9ATSHR
SCHEMBL19853769 0.70 TSHR (0.44) RIPK1ALDH1A1OPRM1OPRL1KMT2A
SCHEMBL19839384 0.69 BLM (0.39) RIPK1ALDH1A1OPRM1OPRL1SMN1; SMN2
SCHEMBL2380442 0.69 SIGMAR1 (0.49) RIPK1ALDH1A1OPRM1OPRL1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018026763-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2018-02-08 WO disclosed