SCHEMBL19856917

SCHEMBL19856917

CC(C)(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)c1cc(C(F)(F)F)ccc1Cl.COc1cc(C)ccc1C(=O)N1C[C@@H]2C[C@H]1CN2C(=O)[C@@H](NC(=O)c1cc2ccccc2[nH]1)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
CTNNB1 P35222 2/20 0.34
DRD4 P21917 3/20 0.33
DRD3 P35462 3/20 0.33
DRD2 P14416 2/20 0.33
HTR1A P08908 2/20 0.33
HTR2A P28223 1/20 0.33
STAT6 P42226 1/20 0.33
CTSA P10619 1/20 0.33
SMYD3 Q9H7B4 1/20 0.33
MCHR1 Q99705 1/20 0.33
ESR1 P03372 1/20 0.33
SCN8A Q9UQD0 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33
CRHR1 P34998 1/20 0.32
CYP51A1 Q16850 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19856946 0.91 DRD2 (0.38) HCRTR1HCRTR2DRD4DRD3DRD2
SCHEMBL19856948 0.91 DRD2 (0.38) HCRTR1HCRTR2DRD4DRD3DRD2
SCHEMBL19856978 0.91 DRD2 (0.39) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL19856980 0.91 DRD2 (0.39) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL19856912 0.87 ESR1 (0.40) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL19856911 0.87 ESR1 (0.40) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL19856959 0.86 ALOX15 (0.40) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL19856908 0.86 ALOX15 (0.40) DRD4DRD3DRD2HTR1AHTR2A
SCHEMBL19856871 0.85 DRD2 (0.41) DRD2STAT6SMYD3CYP51A1TAS1R3
SCHEMBL19856872 0.85 DRD2 (0.41) DRD2STAT6SMYD3CYP51A1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925857-B1 USE OF TRPV4 ANTAGONISTS TO AMELIORATE HYDROCEPHALUS AND RELATED MATERIALS AND METHODS UNIV INDIANA RES & TECH CORP (US) 2018-02-14 EP claimed