SCHEMBL19857043

SCHEMBL19857043

COc1cc(OC(F)(F)F)ccc1-c1cccc(OCc2ncccn2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSA P10619 3/20 0.51
CYP1A1 P04798 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2E1 P05181 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C8 P10632 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2A6 P11509 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP4B1 P13584 1/20 0.47
CYP2B6 P20813 1/20 0.47
CYP3A5 P20815 1/20 0.47
CYP2A7 P20853 1/20 0.47
CYP3A7 P24462 1/20 0.47
CYP2F1 P24903 1/20 0.47
CYP2C18 P33260 1/20 0.47
CYP2C19 P33261 1/20 0.47
CYP2J2 P51589 1/20 0.47
CYP4F2 P78329 1/20 0.47
CYP4F8 P98187 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19857042 0.86 PDE4A (0.45) CYP1A2DYRK1APDE4BPDE4APDE4C
SCHEMBL16824800 0.85 PDE4A (0.48) CYP1A2DYRK1APDE4BPDE4APDE4C
SCHEMBL19857039 0.80 SCN5A (0.46) CTSADYRK1APDE4BPDE4APDE4C
SCHEMBL16821802 0.79 CTSA (0.42) CTSACYP1A1CYP1A2CYP2E1CYP3A4
SCHEMBL19857041 0.75 PPARD (0.45) CTSADYRK1APDE4BPDE4APDE4C
SCHEMBL16824807 0.74 FFAR4 (0.47) CYP1A2PPARD
SCHEMBL19857040 0.71 PDE4A (0.46) PDE4BPDE4APDE4CPDE4D
SCHEMBL19857045 0.71 PPARD (0.46) SYKPPARD
SCHEMBL6345043 0.71 CRHR1 (0.62) CTSACYP1A1CYP1A2CYP2E1CYP3A4
SCHEMBL16821869 0.70 SYK (0.41) SYKMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092234-B1 FUSED HETEROCYCLIC COMPOUNDS AS ION CHANNEL MODULATORS GILEAD SCIENCES INC (US) 2018-02-14 EP disclosed