SCHEMBL19860063

SCHEMBL19860063

O=C(COC(=O)c1ccccc1)Nc1ccc2cnccc2c1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.64
IMPDH2 P12268 2/20 0.60
ROCK2 O75116 2/20 0.59
ALDH1A1 P00352 1/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
MAPT P10636 1/20 0.56
NTRK1 P04629 1/20 0.55
NTRK2 Q16620 1/20 0.55
PRMT3 O60678 1/20 0.54
TDP1 Q9NUW8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12202000 0.85 NOTUM (0.76) NOTUMIMPDH2ROCK2PRMT3
SCHEMBL19860100 0.83 NOTUM (0.65) NOTUMIMPDH2ROCK2ALDH1A1PRMT3
SCHEMBL4428374 0.83 NOTUM (0.62) NOTUMIMPDH2ROCK2PRMT3
SCHEMBL19860099 0.81 NOTUM (0.64) NOTUMIMPDH2ROCK2PRMT3
SCHEMBL12228153 0.80 NOTUM (0.69) NOTUMIMPDH2MEN1KMT2AMAPT
SCHEMBL19860094 0.80 NOTUM (0.68) NOTUMIMPDH2ROCK2PRMT3
SCHEMBL3111893 0.79 IMPDH2 (0.72) IMPDH2ROCK2ALDH1A1MEN1KMT2A
SCHEMBL3595348 0.79 ROCK2 (0.60) NOTUMIMPDH2ROCK2ALDH1A1MEN1
SCHEMBL24735962 0.79 IMPDH2 (0.69) NOTUMIMPDH2ROCK2ALDH1A1PRMT3
SCHEMBL12228149 0.78 NOTUM (0.72) NOTUMIMPDH2ROCK2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed