SCHEMBL19860099

SCHEMBL19860099

O=C(COCc1ccccc1)Nc1ccc2cnccc2c1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.64
IMPDH2 P12268 3/20 0.62
PRMT3 O60678 1/20 0.60
ROCK2 O75116 9/20 0.57
PTPRC P08575 1/20 0.56
PTPN1 P18031 1/20 0.56
ROCK1 Q13464 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12202000 0.85 NOTUM (0.76) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL24735962 0.84 IMPDH2 (0.69) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL12058848 0.83 POLB (0.65) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL14124411 0.83 PRMT3 (0.59) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL19860096 0.83 NOTUM (0.65) NOTUMIMPDH2PRMT3
SCHEMBL3566775 0.83 PRMT3 (0.72) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL13913488 0.81 ROCK2 (0.65) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL19860063 0.81 NOTUM (0.64) NOTUMIMPDH2PRMT3ROCK2
SCHEMBL2164137 0.81 PRMT3 (0.69) NOTUMIMPDH2PRMT3ROCK2ROCK1
SCHEMBL4553921 0.80 PRMT3 (0.56) NOTUMIMPDH2PRMT3ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890123-B2 6-aminoisoquinoline compounds AERIE PHARMACEUTICALS, INC. (US) 2018-02-13 US disclosed