SCHEMBL19902564

SCHEMBL19902564

Cc1c(F)ccc2cc(C(=O)N[C@H]3CC[C@H](c4n[nH]c(=O)c5ccccc54)CC3)[nH]c12

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.44
SETD2 Q9BYW2 2/20 0.44
NSD2 O96028 1/20 0.44
ROCK2 O75116 1/20 0.42
PARP1 P09874 3/20 0.40
PLA2G7 Q13093 9/20 0.39
MAPK8 P45983 1/20 0.38
PYGL P06737 1/20 0.37
PYGM P11217 1/20 0.37
MLLT1 Q03111 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17452863 0.90 ROCK2 (0.55) SMYD3SETD2NSD2ROCK2PARP1
SCHEMBL19902488 0.88 SMYD3 (0.46) SMYD3SETD2NSD2ROCK2PLA2G7
SCHEMBL19902413 0.86 SMYD3 (0.61) SMYD3SETD2NSD2ROCK2PLA2G7
SCHEMBL19902699 0.84 PLA2G7 (0.53) SMYD3SETD2NSD2ROCK2PLA2G7
SCHEMBL19902711 0.83 PYGL (0.48) SMYD3SETD2NSD2ROCK2PLA2G7
SCHEMBL19902625 0.83 MLLT1 (0.49) SMYD3ROCK2MAPK8PYGLPYGM
SCHEMBL19902581 0.82 SMYD3 (0.46) SMYD3SETD2NSD2ROCK2PLA2G7
SCHEMBL19902463 0.82 SLC2A1 (0.46) SMYD3SETD2NSD2ROCK2PLA2G7
SCHEMBL19902474 0.82 PLA2G7 (0.43) SMYD3SETD2NSD2ROCK2PLA2G7
SCHEMBL19902458 0.81 SCN4A (0.48) SMYD3ROCK2MAPK8PYGLPYGM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180155296-A1 SPIROCYCLOHEPTANES AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2018-06-07 US disclosed
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180155296-A1 SPIROCYCLOHEPTANES AS INHIBITORS OF ROCK ROCK1, MYLK, ROCK2 SMYD3 1799/4885SETD2 3022/4885NSD2 3357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.