SCHEMBL19902463

SCHEMBL19902463

O=C(N[C@H]1CC[C@H](c2n[nH]c(=O)c3ccccc32)CC1)c1cc2cccc(C(F)(F)F)c2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.46
SMYD3 Q9H7B4 2/20 0.44
NSD2 O96028 1/20 0.42
SETD2 Q9BYW2 1/20 0.42
PLA2G7 Q13093 9/20 0.41
HRH4 Q9H3N8 2/20 0.40
ROCK2 O75116 1/20 0.39
MAPK8 P45983 1/20 0.38
PTGES O14684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17452844 0.90 ROCK2 (0.51) SLC2A1SMYD3NSD2SETD2PLA2G7
SCHEMBL19902488 0.88 SMYD3 (0.46) SMYD3NSD2SETD2PLA2G7HRH4
SCHEMBL19902699 0.87 PLA2G7 (0.53) SMYD3NSD2SETD2PLA2G7ROCK2
SCHEMBL19902413 0.86 SMYD3 (0.61) SMYD3NSD2SETD2PLA2G7HRH4
SCHEMBL19902711 0.86 PYGL (0.48) SMYD3NSD2SETD2PLA2G7ROCK2
SCHEMBL19902581 0.84 SMYD3 (0.46) SMYD3NSD2SETD2PLA2G7HRH4
SCHEMBL19902458 0.83 SCN4A (0.48) SLC2A1SMYD3ROCK2MAPK8
SCHEMBL19902564 0.82 SMYD3 (0.44) SMYD3NSD2SETD2PLA2G7ROCK2
SCHEMBL19902628 0.81 RIPK1 (0.48) SMYD3PLA2G7HRH4ROCK2MAPK8
SCHEMBL19902412 0.80 ROCK2 (0.43) SMYD3NSD2SETD2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180155296-A1 SPIROCYCLOHEPTANES AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2018-06-07 US disclosed
US-9902702-B2 Spirocycloheptanes as inhibitors of rock BRISTOL-MYERS SQUIBB COMPANY (US) 2018-02-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180155296-A1 SPIROCYCLOHEPTANES AS INHIBITORS OF ROCK ROCK1, MYLK, ROCK2 SLC2A1 3585/4885SMYD3 1799/4885NSD2 3357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.