SCHEMBL19902755

SCHEMBL19902755

CCc1cnccc1C(=N)Nc1ccc(C)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.43
TP53 P04637 3/20 0.42
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
ALDH1A1 P00352 2/20 0.40
NAMPT P43490 2/20 0.40
HSD17B10 Q99714 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
BRAF P15056 1/20 0.39
KDM4E B2RXH2 1/20 0.39
SLC2A1 P11166 2/20 0.39
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19902756 0.90 BLM (0.42) NPC1RAB9ANAMPTMAPTBRAF
SCHEMBL19902783 0.73 SGMS2 (0.35) KMT2ATP53NPC1RAB9AALDH1A1
SCHEMBL19902767 0.71 RAB9A (0.44) NPC1RAB9ANAMPTSMN1; SMN2POLB
SCHEMBL16489237 0.70 MEN1 (0.45) KMT2ANPC1RAB9AALDH1A1NAMPT
SCHEMBL5172599 0.69 KMT2A (0.68) KMT2ATP53NPC1RAB9AALDH1A1
SCHEMBL4480018 0.69 LMNA (0.48) KMT2ATP53NPC1RAB9AALDH1A1
SCHEMBL9192271 0.68 MEN1 (0.73) KMT2ATP53NPC1RAB9AALDH1A1
SCHEMBL16491933 0.68 NPC1 (0.44) KMT2ANPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL25668722 0.67 KMT2A (0.69) KMT2ATP53RAB9AALDH1A1SMN1; SMN2
SCHEMBL13962554 0.66 KMT2A (0.59) KMT2ATP53NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3033337-B1 SUBSTITUTED IMIDAZOLES AS N-TYPE CALCIUM CHANNEL BLOCKERS JANSSEN PHARMACEUTICA NV (BE) 2018-02-28 EP disclosed