SCHEMBL19902763

SCHEMBL19902763

CCc1ccccc1C(=N)Nc1cnc(C)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SGMS2 Q8NHU3 3/20 0.40
HTT P42858 1/20 0.38
F2R P25116 1/20 0.37
CXCR2 P25025 2/20 0.35
HSD17B10 Q99714 3/20 0.35
MAPT P10636 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 2/20 0.35
TP53 P04637 2/20 0.35
RAB9A P51151 2/20 0.35
MAPK1 P28482 2/20 0.35
KDR P35968 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
KCNK3 O14649 1/20 0.34
KCNK9 Q9NPC2 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19902764 0.86 NPSR1 (0.46) SGMS2HTTHSD17B10MAPTNPSR1
SCHEMBL11452798 0.83 NPC1 (0.48) HTTHSD17B10MAPTSMN1; SMN2NPC1
SCHEMBL16491931 0.79 RAB9A (0.44) HSD17B10MAPTNPSR1SMN1; SMN2NPC1
SCHEMBL19902737 0.77 RAB9A (0.54) HTTMAPTNPSR1SMN1; SMN2NPC1
SCHEMBL28858026 0.74 RAB9A (0.40) MAPTSMN1; SMN2NPC1RAB9AKDR
SCHEMBL5763437 0.72 CLCN2 (0.41) HTTF2RMAPTSMN1; SMN2NPC1
SCHEMBL6961935 0.71 GAA (0.46) HTTF2RMAPTHPGDALDH1A1
SCHEMBL19902804 0.70 BLM (0.39) F2RMAPTHPGDALDH1A1GAA
SCHEMBL19902767 0.70 RAB9A (0.44) NPSR1SMN1; SMN2NPC1RAB9A
SCHEMBL459529 0.67 P4HTM (0.42) MAPTSMN1; SMN2NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3033337-B1 SUBSTITUTED IMIDAZOLES AS N-TYPE CALCIUM CHANNEL BLOCKERS JANSSEN PHARMACEUTICA NV (BE) 2018-02-28 EP disclosed