SCHEMBL19904512

SCHEMBL19904512

O=C(NC(Cc1cc(F)c2c(c1)OCCO2)CN1CCC1)[C@@H]1CCN(c2ccc3cc(Cl)sc3c2)C1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.35
NOTUM Q6P988 3/20 0.33
TACR2 P21452 2/20 0.33
PROKR2 Q8NFJ6 2/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
ACACB O00763 2/20 0.31
TRPV1 Q8NER1 1/20 0.31
UGCG Q16739 2/20 0.31
CHRM2 P08172 2/20 0.31
CHRM1 P11229 1/20 0.31
SSTR3 P32745 2/20 0.31
SSTR1 P30872 1/20 0.31
KDM4E B2RXH2 1/20 0.30
HDAC4 P56524 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19904694 0.99 HTR1A (0.35) HTR1ANOTUMTACR2PROKR2PDCD1
SCHEMBL19904590 0.89 KMT2A (0.36) HTR1ANOTUMPROKR2PDCD1CD274
SCHEMBL19904455 0.89 KMT2A (0.36) HTR1ANOTUMPROKR2PDCD1CD274
SCHEMBL19904570 0.88 NAMPT (0.33) HTR1ANOTUMPDCD1CD274ACACB
SCHEMBL19904686 0.88 NAMPT (0.33) HTR1ANOTUMPDCD1CD274ACACB
SCHEMBL19904493 0.88 KMT2A (0.38) HTR1ATACR2PDCD1CD274ACACB
SCHEMBL19904685 0.88 KMT2A (0.38) HTR1ATACR2PDCD1CD274ACACB
SCHEMBL19904488 0.88 KMT2A (0.38) HTR1ANOTUMPROKR2PDCD1CD274
SCHEMBL19904593 0.87 MCHR1 (0.36) HTR1ACHRM2HDAC4
SCHEMBL19904324 0.87 KDM4E (0.37) HTR1ANOTUMACACBTRPV1UGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-B1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARM INC (US) 2018-02-28 EP disclosed